SCHEMBL1913652

SCHEMBL1913652

O=c1ccn(OCCCCCCCCCCF)c(=O)[nH]1

nearest known ligand 0.38

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DUT P33316 7/20 0.38
CRBN Q96SW2 3/20 0.37
L3MBTL1 Q9Y468 1/20 0.35
PKM P14618 1/20 0.35
DDB1 Q16531 1/20 0.34
PDE3A Q14432 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7614894 0.73 PKM (0.51) DUTCRBNL3MBTL1PKMDDB1
SCHEMBL11666542 0.69 CRBN (0.52) DUTCRBNL3MBTL1PKMDDB1
SCHEMBL4409228 0.69 ALDH1A1 (0.41) DUTCRBNL3MBTL1PKMDDB1
SCHEMBL3235869 0.67 L3MBTL1 (0.53) DUTCRBNL3MBTL1PKM
SCHEMBL10618034 0.66 PKM (0.51) DUTCRBNL3MBTL1PKMDDB1
SCHEMBL572752 0.66 CRBN (0.54) DUTCRBNL3MBTL1PKMDDB1
SCHEMBL1913656 0.66
SCHEMBL5705360 0.65 CRBN (0.47) DUTCRBNL3MBTL1PKMDDB1
SCHEMBL6102943 0.64 CRBN (0.56) DUTCRBNL3MBTL1PKMDDB1
SCHEMBL426038 0.64 CRBN (0.45) DUTCRBNL3MBTL1PKMDDB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8921304-B2 Modified ubiquitin proteins having a specific binding activity for the extradomain B of fibronectin SCIL PROTEINS GMBH 2014-12-30 US claimed
EP-2367843-B1 MODIFIED UBIQUITIN PROTEINS HAVING A SPECIFIC BINDING ACTIVITY FOR THE EXTRADOMAIN B OF FIBRONECTIN SCIL PROTEINS GMBH (DE) 2014-10-08 EP claimed
EP-2513138-B1 MODIFIED UBIQUITIN PROTEINS HAVING A SPECIFIC BINDING ACTIVITY FOR THE EXTRADOMAIN B OF FIBRONECTIN SCIL PROTEINS GMBH (DE) 2014-10-01 EP claimed
US-20130011334-A1 MODIFIED UBIQUITIN PROTEINS HAVING A SPECIFIC BINDING ACTIVITY FOR THE EXTRADOMAIN B OF FIBRONECTIN NAVIGO PROTEINS GMBH (DE) 2013-01-10 US claimed
US-20120301393-A1 MODIFIED UBIQUITIN PROTEINS HAVING A SPECIFIC BINDING ACTIVITY FOR THE EXTRADOMAIN B OF FIBRONECTIN SCIL PROTEINS GMBH 2012-11-29 US claimed
EP-2513138-A1 MODIFIED UBIQUITIN PROTEINS HAVING A SPECIFIC BINDING ACTIVITY FOR THE EXTRADOMAIN B OF FIBRONECTIN Scil Proteins GmbH (DE) 2012-10-24 EP claimed
EP-2367843-A1 MODIFIED UBIQUITIN PROTEINS HAVING A SPECIFIC BINDING ACTIVITY FOR THE EXTRADOMAIN B OF FIBRONECTIN Scil Proteins GmbH (DE) 2011-09-28 EP claimed
WO-2011073208-A9 MODIFIED UBIQUITIN PROTEINS HAVING A SPECIFIC BINDING ACTIVITY FOR THE EXTRADOMAIN B OF FIBRONECTIN SCIL PROTEINS GMBH (DE) 2011-08-04 WO claimed
WO-2011073208-A1 MODIFIED UBIQUITIN PROTEINS HAVING A SPECIFIC BINDING ACTIVITY FOR THE EXTRADOMAIN B OF FIBRONECTIN SCIL PROTEINS GMBH (DE) 2011-06-23 WO claimed
WO-2011073209-A1 MODIFIED UBIQUITIN PROTEINS HAVING A SPECIFIC BINDING ACTIVITY FOR THE EXTRADOMAIN B OF FIBRONECTIN SCIL PROTEINS GMBH (DE) 2011-06-23 WO claimed
US-20150183846-A1 HUMAN FUSION PROTEINS COMPRISING SINGLE CHAIN TNFALPHA AND TARGETING DOMAINS SCIL PROTEINS GMBH (DE) 2015-07-02 US disclosed
EP-2861616-A1 HUMAN FUSION PROTEINS COMPRISING SINGLE CHAIN TNFALPHA AND TARGETING DOMAINS Scil Proteins GmbH (DE) 2015-04-22 EP disclosed
US-8921304-B2 Modified ubiquitin proteins having a specific binding activity for the extradomain B of fibronectin SCIL PROTEINS GMBH 2014-12-30 US disclosed
EP-2367843-B1 MODIFIED UBIQUITIN PROTEINS HAVING A SPECIFIC BINDING ACTIVITY FOR THE EXTRADOMAIN B OF FIBRONECTIN SCIL PROTEINS GMBH (DE) 2014-10-08 EP disclosed
EP-2513138-B1 MODIFIED UBIQUITIN PROTEINS HAVING A SPECIFIC BINDING ACTIVITY FOR THE EXTRADOMAIN B OF FIBRONECTIN SCIL PROTEINS GMBH (DE) 2014-10-01 EP disclosed
EP-2513138-A1 MODIFIED UBIQUITIN PROTEINS HAVING A SPECIFIC BINDING ACTIVITY FOR THE EXTRADOMAIN B OF FIBRONECTIN Scil Proteins GmbH (DE) 2012-10-24 EP disclosed
EP-2367843-A1 MODIFIED UBIQUITIN PROTEINS HAVING A SPECIFIC BINDING ACTIVITY FOR THE EXTRADOMAIN B OF FIBRONECTIN Scil Proteins GmbH (DE) 2011-09-28 EP disclosed
WO-2011073208-A9 MODIFIED UBIQUITIN PROTEINS HAVING A SPECIFIC BINDING ACTIVITY FOR THE EXTRADOMAIN B OF FIBRONECTIN SCIL PROTEINS GMBH (DE) 2011-08-04 WO disclosed
WO-2011073208-A1 MODIFIED UBIQUITIN PROTEINS HAVING A SPECIFIC BINDING ACTIVITY FOR THE EXTRADOMAIN B OF FIBRONECTIN SCIL PROTEINS GMBH (DE) 2011-06-23 WO disclosed
WO-2011073209-A1 MODIFIED UBIQUITIN PROTEINS HAVING A SPECIFIC BINDING ACTIVITY FOR THE EXTRADOMAIN B OF FIBRONECTIN SCIL PROTEINS GMBH (DE) 2011-06-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120301393-A1 MODIFIED UBIQUITIN PROTEINS HAVING A SPECIFIC BINDING ACTIVITY FOR THE EXTRADOMAIN B OF FIBRONECTIN STUB1, UBE4A, UBE2B DUT 1855/4885CRBN 243/4885L3MBTL1 2622/4885
US-20130011334-A1 MODIFIED UBIQUITIN PROTEINS HAVING A SPECIFIC BINDING ACTIVITY FOR THE EXTRADOMAIN B OF FIBRONECTIN STUB1, UBE2B, UBE4A DUT 2522/4885CRBN 206/4885L3MBTL1 2574/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.