SCHEMBL19141069

SCHEMBL19141069

O=C(NS)c1cc(Cl)ccc1O

nearest known ligand 0.64

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
P2RX1 P51575 9/20 0.64
KCNMA1 Q12791 5/20 0.64
TMPRSS4 Q9NRS4 6/20 0.62
P2RX4 Q99571 5/20 0.62
P2RX7 Q99572 5/20 0.62
CA1 P00915 1/20 0.60
CA2 P00918 1/20 0.60
CDK1 P06493 1/20 0.57
TAS1R3 Q7RTX0 1/20 0.53
TAS1R1 Q7RTX1 1/20 0.53
TAS1R2 Q8TE23 1/20 0.53
MEN1 O00255 1/20 0.53
IKBKB O14920 1/20 0.53
CHUK O15111 1/20 0.53
KDR P35968 1/20 0.53
FLT3 P36888 1/20 0.53
KMT2A Q03164 1/20 0.53
MYLK Q15746 1/20 0.53
MAP4K5 Q9Y4K4 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11324189 0.84 P2RX1 (0.68) P2RX1KCNMA1TMPRSS4P2RX4P2RX7
SCHEMBL5506621 0.82 P2RX1 (0.66) P2RX1KCNMA1TMPRSS4P2RX4P2RX7
SCHEMBL3871841 0.81 P2RX1 (0.64) P2RX1KCNMA1TMPRSS4P2RX4P2RX7
SCHEMBL3277584 0.81 ALDH1A1 (0.70) P2RX1KCNMA1TMPRSS4P2RX4P2RX7
SCHEMBL2169619 0.78 P2RX1 (1.00) P2RX1KCNMA1TMPRSS4P2RX4P2RX7
SCHEMBL29454776 0.78 P2RX1 (1.00) P2RX1KCNMA1TMPRSS4P2RX4P2RX7
SCHEMBL6401690 0.78 CA1 (0.67) P2RX1KCNMA1TMPRSS4P2RX4P2RX7
SCHEMBL6966672 0.77 CA1 (0.72) P2RX1KCNMA1TMPRSS4P2RX4P2RX7
SCHEMBL21423064 0.77 ALOX5 (0.66) P2RX1KCNMA1TMPRSS4P2RX4P2RX7
SCHEMBL27786747 0.77 TMPRSS4 (0.60) P2RX1KCNMA1TMPRSS4P2RX4P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3192794-A1 SUSTAINED HIV PROTEASE INHIBITOR Shionogi & Co., Ltd. (JP) 2017-07-19 EP disclosed