SCHEMBL19174286

SCHEMBL19174286

Oc1ccc(F)cc1CCCCCNC[C@H](O)CCCc1cc(F)ccc1O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 11/20 0.45
ADRB1 P08588 7/20 0.43
MPO P05164 5/20 0.40
ADRB3 P13945 5/20 0.39
SLC6A4 P31645 3/20 0.39
KDM4E B2RXH2 1/20 0.39
HTR1A P08908 1/20 0.39
CHRM5 P08912 1/20 0.39
DRD2 P14416 1/20 0.39
ADRA2B P18089 1/20 0.39
DRD4 P21917 1/20 0.39
SLC6A2 P23975 1/20 0.39
FPR3 P25089 1/20 0.39
ADRA1D P25100 1/20 0.39
HTR1D P28221 1/20 0.39
HTR1B P28222 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
GPR183 P32249 1/20 0.39
HTR7 P34969 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19174337 1.00 ADRB2 (0.45) ADRB2ADRB1MPOADRB3SLC6A4
SCHEMBL15107034 0.91 MPO (0.43) ADRB2ADRB1MPOADRB3SLC6A4
SCHEMBL6857021 0.81 MPO (0.48) ADRB2ADRB1MPOADRB3SLC6A4
SCHEMBL17011674 0.80 ACLY (0.35) MPOSLC6A4HTR1AKCNH2TMEM97
SCHEMBL17011675 0.80 ACLY (0.35) MPOSLC6A4HTR1AKCNH2TMEM97
SCHEMBL23940684 0.79 ACLY (0.36) ADRB2ADRB1MPOSLC6A4HTR1A
SCHEMBL12397446 0.79 ACLY (0.36) ADRB2ADRB1MPOSLC6A4HTR1A
SCHEMBL18697459 0.79 ACLY (0.36) ADRB2ADRB1MPOSLC6A4HTR1A
SCHEMBL19174208 0.75 MPO (0.63) MPOSLC6A4CA12CA2CA9
SCHEMBL14240235 0.72 ADRB2 (0.68) ADRB2ADRB1ADRB3SLC6A4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3405467-B1 PROCESS FOR THE SYNTHESIS OF INTERMEDIATES OF NEBIVOLOL MENARINI INT OPERATIONS LUXEMBOURG SA (LU) 2021-08-04 EP disclosed
WO-2017125900-A1 PROCESS FOR THE SYNTHESIS OF INTERMEDIATES OF NEBIVOLOL MENARINI INTERNATIONAL OPERATIONS LUXEMBOURG S.A. (LU) 2017-07-27 WO disclosed