SCHEMBL19185358

SCHEMBL19185358

CC(C)(C)c1ncnc2[nH]cc(F)c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 3/20 0.41
TRPA1 O75762 4/20 0.38
LRRK2 Q5S007 6/20 0.38
PRKD3 O94806 1/20 0.38
MAP4K4 O95819 1/20 0.38
PAK4 O96013 1/20 0.38
NTRK1 P04629 1/20 0.38
PRKACA P17612 1/20 0.38
LTK P29376 1/20 0.38
MAP2K2 P36507 1/20 0.38
MAPK8 P45983 1/20 0.38
CDK8 P49336 1/20 0.38
CLK2 P49760 1/20 0.38
GSK3A P49840 1/20 0.38
GSK3B P49841 1/20 0.38
RPS6KA3 P51812 1/20 0.38
CDK5 Q00535 1/20 0.38
MAP2K1 Q02750 1/20 0.38
PRKCQ Q04759 1/20 0.38
MST1R Q04912 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17032328 0.81 AKT1 (0.42) IRAK4TRPA1LRRK2PRKD3MAP4K4
SCHEMBL19185239 0.77 MAP3K7 (0.54) IRAK4LRRK2ROCK1MAP3K7TAB1
SCHEMBL19185382 0.75 MAP3K7 (0.41) MAP3K7TAB1JAK2JAK3
SCHEMBL14649091 0.75 TRPA1 (0.44) IRAK4TRPA1LRRK2CHEK1BRAF
SCHEMBL27050490 0.73 LRRK2 (0.31) LRRK2
SCHEMBL6531144 0.72 RET (0.42) IRAK4TRPA1LRRK2CHEK1BRAF
SCHEMBL14667020 0.71 GPR84 (0.32) TRPA1
SCHEMBL153752 0.71 CHEK1 (0.63) IRAK4TRPA1LRRK2DYRK1ACHEK1
SCHEMBL18868081 0.70 IRAK4 (0.41) IRAK4TRPA1LRRK2CHEK1BRAF
SCHEMBL24656161 0.69 JAK2 (0.38) IRAK4LRRK2CDK5ROCK1JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9718815-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2017-08-01 US disclosed