SCHEMBL19202673

SCHEMBL19202673

N=Cc1cc(C2CCN(C=O)CC2)nc(-c2ccc(CN3CCCC3)cc2)c1N

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.44
DRD4 P21917 2/20 0.44
DRD3 P35462 2/20 0.44
DCTPP1 Q9H773 4/20 0.40
ADORA2A P29274 2/20 0.39
ADORA1 P30542 2/20 0.39
ATR Q13535 1/20 0.38
BTK Q06187 1/20 0.37
AKT1 P31749 6/20 0.37
AKT2 P31751 6/20 0.37
AKT3 Q9Y243 1/20 0.37
CXCR3 P49682 1/20 0.36
DAGLA Q9Y4D2 1/20 0.35
HRH3 Q9Y5N1 2/20 0.35
HRH4 Q9H3N8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19202672 0.84 BTK (0.50) DRD2DRD4DRD3BTKHRH3
SCHEMBL24083375 0.79 BTK (0.57) DRD2DRD4DRD3DCTPP1ATR
SCHEMBL24083366 0.73 BTK (0.70) BTK
SCHEMBL24083370 0.72 BTK (0.51) BTK
SCHEMBL24083387 0.71 BTK (0.46) BTK
SCHEMBL24083393 0.64 TNK2 (0.45) BTK
SCHEMBL24083385 0.64 BTK (0.41) BTK
SCHEMBL24083394 0.64 BTK (0.52) BTK
SCHEMBL6975763 0.62 DRD2 (0.86) DRD2DRD4DRD3ADORA2AADORA1
SCHEMBL1387890 0.61 DRD4 (1.00) DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017128917-A1 PARAZOLE CONDENSED-RING DERIVATIVES AND PREPARATION METHOD THEREOF AND APPLICATION THEREOF IN TREATMENT OF CANCERS, INFLAMMATION AND IMMUNE DISEASES 北京诺诚健华医药科技有限公司 2017-08-03 WO disclosed