SCHEMBL1922545

SCHEMBL1922545

COc1cc(C)c(CCCO)cn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NNMT P40261 1/20 0.45
GCK P35557 2/20 0.37
CYP2A6 P11509 1/20 0.36
FFAR1 O14842 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36
MTNR1A P48039 2/20 0.34
MTNR1B P49286 2/20 0.34
DHFR P00374 2/20 0.33
HSP90AA1 P07900 1/20 0.33
MEN1 O00255 1/20 0.33
PABPC1 P11940 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B1 P14061 1/20 0.33
HSD17B2 P37059 1/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
CYP11B1 P15538 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22145148 0.82 NNMT (0.50) NNMTCYP2A6DHFRMEN1PABPC1
SCHEMBL20095717 0.81 FFAR1 (0.48) NNMTFFAR1MEN1KMT2A
SCHEMBL18396986 0.79 NNMT (0.44) NNMTCYP2A6FFAR1MTNR1AMTNR1B
SCHEMBL2542011 0.79 MTNR1A (0.36) NNMTGCKTNKS2MTNR1AMTNR1B
SCHEMBL10263430 0.77 NOS3 (0.55) NNMTCYP2A6DHFRMEN1PABPC1
SCHEMBL29863385 0.77 HTR2A (0.41) NNMTMTNR1AMTNR1BNOS1
SCHEMBL21459468 0.77 HTR2A (0.41) NNMTMTNR1AMTNR1BNOS1
SCHEMBL22145202 0.75 NNMT (0.46) NNMTCYP2A6DHFRMEN1PABPC1
SCHEMBL30987534 0.75 NNMT (0.46) NNMTCYP2A6DHFRMEN1PABPC1
SCHEMBL21327094 0.75 NNMT (0.50) NNMTCYP2A6FFAR1DHFRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2328902-A1 PYRAZOLO [5,1-B]OXAZOLE DERIVATIVES AS CRF1 ANTAGONISTS Novartis AG (CH) 2011-06-08 EP disclosed
WO-2010015628-A1 PYRAZOLO [5,1-B] OXAZOLE DERIVATIVES AS CRF1 ANTAGONISTS NOVARTIS AG (CH) 2010-02-11 WO disclosed