SCHEMBL22145202

SCHEMBL22145202

COc1cc(C)c(CBr)cn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NNMT P40261 1/20 0.46
CYP2A6 P11509 1/20 0.40
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
NOS2 P35228 1/20 0.36
DHFR P00374 3/20 0.36
LOX P28300 1/20 0.34
LOXL2 Q9Y4K0 1/20 0.34
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 2/20 0.33
MEN1 O00255 1/20 0.33
PABPC1 P11940 1/20 0.33
KMT2A Q03164 1/20 0.33
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB1 P18505 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA5 P31644 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18396986 0.85 NNMT (0.44) NNMTCYP2A6NOS3NOS1NOS2
SCHEMBL26144367 0.85 NNMT (0.42) NNMTCYP2A6DHFRLOXLOXL2
SCHEMBL10263430 0.82 NOS3 (0.55) NNMTCYP2A6NOS3NOS1NOS2
SCHEMBL6794136 0.81 TUBB4A (0.39) NNMTLOXLOXL2SLC6A2SLC6A4
SCHEMBL30987534 0.81 NNMT (0.46) NNMTCYP2A6NOS3NOS1NOS2
SCHEMBL22145148 0.81 NNMT (0.50) NNMTCYP2A6NOS3NOS1NOS2
SCHEMBL21327094 0.81 NNMT (0.50) NNMTCYP2A6NOS3NOS1NOS2
SCHEMBL22122764 0.79 HTR1A (0.34) NNMTDHFRLOXLOXL2GABRP
SCHEMBL9013521 0.77 NNMT (0.35) NNMTLOXLOXL2MEN1KMT2A
SCHEMBL30486638 0.77 NNMT (0.35) NNMTLOXLOXL2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020127508-A1 SUBSTITUTED OXOPYRIDINE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2020-06-25 WO disclosed