SCHEMBL1922840

SCHEMBL1922840

CCc1cnc(N2CCC(CCCOc3ccc(N4CCNC(=O)C4)nc3)CC2)nc1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 13/20 0.47
HPGDS O60760 1/20 0.40
LRRK2 Q5S007 2/20 0.37
CYP4F2 P78329 1/20 0.37
CYP4A11 Q02928 1/20 0.37
KCNH2 Q12809 1/20 0.37
ACACB O00763 1/20 0.37
PRMT5 O14744 1/20 0.36
LCAT P04180 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13534680 0.85 HPGDS (0.44) GPR119HPGDSLRRK2CYP4F2CYP4A11
SCHEMBL1922669 0.77 GPR119 (0.52) GPR119KCNH2
SCHEMBL26944604 0.76 HPGDS (0.45) GPR119HPGDSLRRK2PRMT5LCAT
SCHEMBL3189635 0.72 GPR119 (0.50) GPR119KCNH2
SCHEMBL11956888 0.71 GPR119 (0.53) GPR119ACACB
SCHEMBL29892851 0.71 GPR119 (0.57) GPR119KCNH2
SCHEMBL1295470 0.71 GPR119 (0.49) GPR119CYP4F2CYP4A11KCNH2
SCHEMBL1924194 0.71 GPR119 (0.54) GPR119
SCHEMBL12356451 0.70 GPR119 (0.53) GPR119
SCHEMBL1295887 0.70 GPR119 (0.48) GPR119KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110212939-A1 Heterocyclic GPCR Agonists PROSIDION LIMITED (GB) 2011-09-01 US disclosed
US-20110212939-A1 Heterocyclic GPCR Agonists PROSIDION LIMITED (GB) 2011-09-01 US disclosed
US-20110212939-A1 Heterocyclic GPCR Agonists PROSIDION LIMITED (GB) 2011-09-01 US disclosed
EP-2328867-A1 HETEROCYCLIC GPCR AGONISTS Prosidion Limited (GB) 2011-06-08 EP disclosed
WO-2010004347-A1 HETEROCYCLIC GPCR AGONISTS PROSIDION LIMITED (GB) 2010-01-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110212939-A1 Heterocyclic GPCR Agonists GPR119, GCGR, GPR27 GPR119 1/4885HPGDS 1166/4885LRRK2 930/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.