SCHEMBL19230285

SCHEMBL19230285

Oc1ccc(C2CCc3cc(Br)ccc3O2)c(Cl)c1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 9/20 0.57
ESR1 P03372 9/20 0.57
AR P10275 1/20 0.40
TTR P02766 1/20 0.36
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
CYP19A1 P11511 1/20 0.34
TYR P14679 1/20 0.34
PDK1 Q15118 1/20 0.34
PDK2 Q15119 1/20 0.34
PDK3 Q15120 1/20 0.34
PDK4 Q16654 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19230670 0.90 ESR2 (0.53) ESR2ESR1
SCHEMBL4366876 0.85 ESR2 (0.61) ESR2ESR1ARTTRPTGS1
SCHEMBL19230545 0.81 ESR1 (0.53) ESR2ESR1TTRCYP19A1
SCHEMBL28649906 0.81 ESR1 (0.53) ESR2ESR1ARTTRPDK1
SCHEMBL19230953 0.81 ESR2 (0.50) ESR2ESR1ARPDK1PDK2
SCHEMBL4371924 0.81 ESR2 (0.62) ESR2ESR1ARTTRCYP19A1
SCHEMBL4368187 0.79 ESR2 (0.68) ESR2ESR1ARCYP19A1
SCHEMBL19230284 0.79 AR (0.66) ESR2ARTTRPTGS1PTGS2
SCHEMBL19230656 0.78 ESR1 (0.49) ESR2ESR1PDK1PDK2PDK3
SCHEMBL19230805 0.78 ESR1 (0.49) ESR2ESR1PDK1PDK2PDK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602811-B FXR receptor agonists 轩竹生物科技有限公司 2021-11-16 CN disclosed
WO-2017133521-A1 FXR RECEPTOR AGONIST 山东轩竹医药科技有限公司 2017-08-10 WO disclosed