SCHEMBL28649906

SCHEMBL28649906

O=C(O)c1ccc2c(c1)CCC(c1ccc(O)cc1Cl)O2

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.53
ESR2 Q92731 4/20 0.53
TDP1 Q9NUW8 1/20 0.44
MCL1 Q07820 4/20 0.44
AR P10275 2/20 0.39
PDK1 Q15118 1/20 0.39
PDK2 Q15119 1/20 0.39
PDK3 Q15120 1/20 0.39
PDK4 Q16654 1/20 0.39
TTR P02766 2/20 0.38
SRD5A1 P18405 1/20 0.37
SRD5A2 P31213 1/20 0.37
CYP3A4 P08684 1/20 0.37
FABP4 P15090 2/20 0.36
NR1H4 Q96RI1 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19230656 0.86 ESR1 (0.49) ESR1ESR2MCL1PDK1PDK2
SCHEMBL19230805 0.86 ESR1 (0.49) ESR1ESR2MCL1PDK1PDK2
SCHEMBL19230310 0.86 ESR1 (0.49) ESR1ESR2MCL1PDK1PDK2
SCHEMBL4366876 0.82 ESR2 (0.61) ESR1ESR2MCL1ARTTR
SCHEMBL19230285 0.81 ESR2 (0.57) ESR1ESR2ARPDK1PDK2
SCHEMBL19230618 0.81 ESR2 (0.72) ESR1ESR2TDP1MCL1AR
SCHEMBL19230545 0.79 ESR1 (0.53) ESR1ESR2TTR
SCHEMBL4371924 0.78 ESR2 (0.62) ESR1ESR2ARTTRCYP3A4
SCHEMBL19230672 0.77 ESR2 (0.46) ESR1ESR2
SCHEMBL19230647 0.74 RAB9A (0.43) TDP1MCL1ARTTRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602811-B FXR receptor agonists 轩竹生物科技有限公司 2021-11-16 CN disclosed