SCHEMBL19230369

SCHEMBL19230369

COC(=O)c1ccc2c(c1)CCC(c1ccc(OC/C(C(=N)c3c(Cl)cccc3Cl)=C(/O)C3CC3)cc1Cl)C2=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 3/20 0.36
ITGA2B P08514 3/20 0.36
FAAH O00519 4/20 0.33
GPR84 Q9NQS5 2/20 0.33
ACHE P22303 2/20 0.32
NR1H4 Q96RI1 1/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
CYP2C19 P33261 1/20 0.32
RECQL P46063 1/20 0.32
KMT2A Q03164 1/20 0.31
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19230756 0.92 ITGB3 (0.38) ITGB3ITGA2BNR1H4NPC1RAB9A
SCHEMBL19230576 0.86 ITGB3 (0.35) ITGB3ITGA2B
SCHEMBL19230320 0.85 FAAH (0.38) ITGB3ITGA2BFAAHKMT2ATAS1R3
SCHEMBL19230598 0.82 FAAH (0.34) FAAHNR1H4LMNATP53ALDH1A1
SCHEMBL19230657 0.79 SLC8A1 (0.36) ITGB3ITGA2B
SCHEMBL19230377 0.79 SLC8A1 (0.37) ITGB3ITGA2BNR1H4
SCHEMBL19230764 0.78 SLC8A1 (0.40)
SCHEMBL19230784 0.77 SLC8A1 (0.36) ITGB3ITGA2B
SCHEMBL19230677 0.76 FAAH (0.35) FAAHRAB9ATAS1R3TAS1R1TAS1R2
SCHEMBL19230512 0.76 NR1H4 (0.37) ITGB3ITGA2BFAAHNR1H4NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017133521-A1 FXR RECEPTOR AGONIST 山东轩竹医药科技有限公司 2017-08-10 WO disclosed