SCHEMBL19230756

SCHEMBL19230756

N=C(/C(COc1ccc(C2CCc3cc(C(=O)O)ccc3C2=O)c(Cl)c1)=C(\O)C1CC1)c1c(Cl)cccc1Cl

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.38
ITGA2B P08514 1/20 0.38
NR1H4 Q96RI1 13/20 0.36
SRD5A2 P31213 2/20 0.35
MRGPRX4 Q96LA9 1/20 0.35
FXR2 P51116 1/20 0.34
NPC1 O15118 1/20 0.33
NR4A2 P43354 1/20 0.33
RAB9A P51151 1/20 0.33
SRD5A1 P18405 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19230369 0.92 ITGB3 (0.36) ITGB3ITGA2BNR1H4NPC1RAB9A
SCHEMBL19230576 0.89 ITGB3 (0.35) ITGB3ITGA2B
SCHEMBL19230512 0.84 NR1H4 (0.37) ITGB3ITGA2BNR1H4MRGPRX4FXR2
SCHEMBL19230827 0.77 NR1H4 (0.37) ITGB3ITGA2BNR1H4
SCHEMBL19620251 0.76 NR1H4 (0.40) NR1H4MRGPRX4FXR2
SCHEMBL19230696 0.76 ITGB3 (0.39) ITGB3ITGA2BNR1H4
SCHEMBL19230320 0.76 FAAH (0.38) ITGB3ITGA2B
SCHEMBL19230560 0.76 NR1H4 (0.37) ITGB3ITGA2BNR1H4MRGPRX4
SCHEMBL19230633 0.76 MRGPRX4 (0.38) ITGB3ITGA2BNR1H4MRGPRX4
SCHEMBL20094741 0.75 OPRD1 (0.35) NR1H4MRGPRX4NPC1NR4A2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017133521-A1 FXR RECEPTOR AGONIST 山东轩竹医药科技有限公司 2017-08-10 WO disclosed