SCHEMBL19230647

SCHEMBL19230647

COC(=O)c1ccc2c(c1)CC(c1ccc(O)cc1Cl)O2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.43
CHRNB2 P17787 1/20 0.41
CHRNA4 P43681 1/20 0.41
TDP1 Q9NUW8 1/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
CYP19A1 P11511 1/20 0.39
TYR P14679 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CYP3A4 P08684 1/20 0.38
AR P10275 1/20 0.38
NISCH Q9Y2I1 1/20 0.38
HSP90AA1 P07900 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19230310 0.89 ESR1 (0.49) RAB9ACHRNB2CHRNA4CA12CA1
SCHEMBL19230805 0.89 ESR1 (0.49) RAB9ACHRNB2CHRNA4CA12CA1
SCHEMBL19230656 0.89 ESR1 (0.49) RAB9ACHRNB2CHRNA4CA12CA1
SCHEMBL19230648 0.83 RAB9A (0.42) RAB9ACA12CA1CA2CA7
SCHEMBL19230672 0.82 ESR2 (0.46) CA12CA1CA2CA7CA9
SCHEMBL19230646 0.79 HSD11B1 (0.36) RAB9ACHRNB2CHRNA4TDP1MEN1
SCHEMBL19230623 0.77 ESR1 (0.45) RAB9ACA12CA1CA2CA7
SCHEMBL19230993 0.76 ESR1 (0.47) RAB9ACHRNB2CHRNA4CA12CA1
SCHEMBL19230375 0.76 ESR2 (0.46) RAB9ACHRNB2CHRNA4CA12CA1
SCHEMBL19230316 0.75 CHRNB2 (0.43) CHRNB2CHRNA4CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602811-B FXR receptor agonists 轩竹生物科技有限公司 2021-11-16 CN disclosed
WO-2017133521-A1 FXR RECEPTOR AGONIST 山东轩竹医药科技有限公司 2017-08-10 WO disclosed