SCHEMBL19230697

SCHEMBL19230697

CCOC(=O)c1ccc(OCc2ccccc2)nc1C(F)(F)F

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.51
MEN1 O00255 1/20 0.49
HSP90AA1 P07900 1/20 0.49
KMT2A Q03164 1/20 0.49
GABRA5 P31644 1/20 0.47
NPSR1 Q6W5P4 2/20 0.47
MAOB P27338 1/20 0.45
RAB9A P51151 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
NMT2 O60551 1/20 0.44
NMT1 P30419 1/20 0.44
PPIA P62937 1/20 0.43
TSHR P16473 2/20 0.43
P2RY12 Q9H244 2/20 0.43
ALDH1A1 P00352 2/20 0.42
NPC1 O15118 1/20 0.42
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19230819 0.85 GRM5 (0.42) MAOBRAB9AALDH1A1NPC1NFKB1
SCHEMBL31193929 0.83 KDM4E (0.55) KDM4ENPSR1RAB9AL3MBTL1TSHR
SCHEMBL4126156 0.81 POLB (0.53) KDM4EMEN1HSP90AA1KMT2AGABRA5
SCHEMBL6380407 0.81 KDM4E (0.56) KDM4ENPSR1TSHRALDH1A1NFKB1
SCHEMBL19230699 0.81 PKM (0.42) MAOBL3MBTL1ALDH1A1SMN1; SMN2
SCHEMBL6377043 0.76 KDM4E (0.59) KDM4EMEN1KMT2ANPSR1TSHR
SCHEMBL26641047 0.75 MAPT (0.46) KDM4EMEN1KMT2AGABRA5NPSR1
SCHEMBL5077233 0.75 KDM4E (0.58) KDM4EMEN1HSP90AA1KMT2ANPSR1
SCHEMBL4192553 0.75 KDM4E (0.58) KDM4ENPSR1RAB9ATSHRALDH1A1
SCHEMBL474055 0.74 KDM4E (0.57) KDM4ENPSR1TSHRP2RY12ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602811-B FXR receptor agonists 轩竹生物科技有限公司 2021-11-16 CN disclosed
CN-108602811-A FXR receptor stimulating agents 山东轩竹医药科技有限公司 2018-09-28 CN disclosed
WO-2017133521-A1 FXR RECEPTOR AGONIST 山东轩竹医药科技有限公司 2017-08-10 WO disclosed