SCHEMBL19230699

SCHEMBL19230699

Cc1ccc(OCc2ccccc2)nc1C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.42
GRM5 P41594 2/20 0.42
HTT P42858 2/20 0.42
LMNA P02545 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
NUDT1 P36639 1/20 0.40
STAT3 P40763 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
BRD4 O60885 1/20 0.39
GAA P10253 2/20 0.39
PDE10A Q9Y233 1/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19230697 0.81 KDM4E (0.51) L3MBTL1ALDH1A1SMN1; SMN2MAOB
SCHEMBL22871232 0.80 HPGD (0.39) HTTALDH1A1MAPTMAPK1MAOA
SCHEMBL19230819 0.80 GRM5 (0.42) PKMGRM5HTTALDH1A1MAPT
SCHEMBL19008193 0.80 PKM (0.45) PKMGRM5HTTLMNAL3MBTL1
SCHEMBL19230698 0.79 GRM5 (0.40) PKMGRM5LMNA
SCHEMBL19007909 0.79 L3MBTL1 (0.51) PKMGRM5HTTLMNAL3MBTL1
SCHEMBL19230555 0.78 GRM5 (0.42) PKMGRM5L3MBTL1MAPTSMN1; SMN2
SCHEMBL24461271 0.76 PKM (0.45) PKMGRM5HTTLMNAL3MBTL1
SCHEMBL19273376 0.76 NUDT1 (0.49) PKML3MBTL1ALDH1A1MAPTMAPK1
SCHEMBL24497447 0.76 PKM (0.45) PKMGRM5HTTLMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017133521-A1 FXR RECEPTOR AGONIST 山东轩竹医药科技有限公司 2017-08-10 WO disclosed