SCHEMBL1923699

SCHEMBL1923699

c1ccc(Nc2nc(NCc3cccnc3)nc(Nc3ccccc3)n2)cc1

nearest known ligand 0.73

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNH3 Q9ULD8 6/20 0.73
LTA4H P09960 1/20 0.73
GPR84 Q9NQS5 1/20 0.57
PKM P14618 1/20 0.56
RAD52 P43351 1/20 0.56
ALDH1A1 P00352 2/20 0.54
CYP1A2 P05177 2/20 0.53
CYP2D6 P10635 2/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
KDM4E B2RXH2 1/20 0.53
RECQL P46063 1/20 0.53
MCL1 Q07820 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30784989 0.93 PKM (0.67) KCNH3LTA4HGPR84PKMRAD52
SCHEMBL1923875 0.86 KCNH3 (0.71) KCNH3LTA4HALDH1A1
SCHEMBL523753 0.84 LTA4H (1.00) LTA4HGPR84ALDH1A1CYP1A2CYP2D6
SCHEMBL30642394 0.84 LTA4H (1.00) LTA4HGPR84ALDH1A1CYP1A2CYP2D6
SCHEMBL1924273 0.83 KCNH3 (1.00) KCNH3RECQLMCL1
SCHEMBL5605047 0.79 LTA4H (0.82) LTA4HALDH1A1CYP1A2CYP2D6CYP2C19
SCHEMBL4805011 0.78 LTA4H (0.79) KCNH3LTA4HALDH1A1CYP1A2CYP2D6
SCHEMBL1310247 0.77 PKM (0.76) LTA4HGPR84PKMRAD52ALDH1A1
SCHEMBL30784987 0.77 MEN1 (0.62) LTA4HGPR84PKMRAD52ALDH1A1
SCHEMBL30784980 0.77 MEN1 (0.62) LTA4HGPR84PKMRAD52ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1479397-B1 2,4,6-TRIAMINO-1,3,5-TRIAZINE DERIVATIVE ASTELLAS PHARMA INC (JP) 2011-06-08 EP claimed
US-7375222-B2 2,4,6-Triamino-1,3,5-triazine derivative ASTELLAS PHARMA INC. (JP) 2008-05-20 US claimed