SCHEMBL1923780

SCHEMBL1923780

COc1ccc(Nc2nc(NCc3ccncn3)nc(Nc3ccc(F)cc3)n2)cc1

nearest known ligand 0.81

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNH3 Q9ULD8 14/20 0.81
ALDH1A1 P00352 1/20 0.46
MAPT P10636 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
MEN1 O00255 1/20 0.46
GAA P10253 1/20 0.46
KMT2A Q03164 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
PDE4B Q07343 1/20 0.45
PDE4D Q08499 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1282204 0.90 KCNH3 (1.00) KCNH3
SCHEMBL1923864 0.85 KCNH3 (0.90) KCNH3
SCHEMBL1282182 0.81 KCNH3 (1.00) KCNH3ALDH1A1MAPTNPSR1MEN1
SCHEMBL1923730 0.77 KCNH3 (0.98) KCNH3ALDH1A1MAPTNPSR1MEN1
Hydrochloric Acid SCHEMBL3411999 0.76 KCNH3 (1.00) KCNH3
SCHEMBL5017676 0.75 KCNH3 (0.69) KCNH3ALDH1A1MAPTMEN1GAA
SCHEMBL1924158 0.73 KCNH3 (0.71) KCNH3
SCHEMBL11812041 0.71 MAPT (0.81) KCNH3ALDH1A1MAPTNPSR1MEN1
SCHEMBL1923563 0.71 KCNH3 (0.97) KCNH3
SCHEMBL1391546 0.71 PDE4B (0.70) KCNH3ALDH1A1MAPTNPSR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1479397-B1 2,4,6-TRIAMINO-1,3,5-TRIAZINE DERIVATIVE ASTELLAS PHARMA INC (JP) 2011-06-08 EP claimed
US-7375222-B2 2,4,6-Triamino-1,3,5-triazine derivative ASTELLAS PHARMA INC. (JP) 2008-05-20 US claimed