SCHEMBL1282182

SCHEMBL1282182

COc1ccc(Nc2nc(NCc3ncccn3)nc(Nc3ccc(F)cc3)n2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH3 Q9ULD8 14/20 1.00
ALDH1A1 P00352 2/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
MAPT P10636 2/20 0.50
GAA P10253 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
MAPK1 P28482 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
EGFR P00533 1/20 0.50
PDE4B Q07343 1/20 0.49
PDE4D Q08499 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1280999 0.89 KCNH3 (1.00) KCNH3
SCHEMBL535908 0.85 KCNH3 (1.00) KCNH3
SCHEMBL540957 0.83 KCNH3 (0.86) KCNH3ALDH1A1SMN1; SMN2MAPK1
SCHEMBL1923730 0.81 KCNH3 (0.98) KCNH3ALDH1A1MEN1KMT2AMAPT
SCHEMBL1923780 0.81 KCNH3 (0.81) KCNH3ALDH1A1MEN1KMT2AMAPT
Hydrochloric Acid SCHEMBL3411999 0.80 KCNH3 (1.00) KCNH3
SCHEMBL5017676 0.79 KCNH3 (0.69) KCNH3ALDH1A1MEN1KMT2AMAPT
SCHEMBL1923771 0.76 KCNH3 (0.82) KCNH3MEN1KMT2AMAPTGAA
SCHEMBL11812041 0.75 MAPT (0.81) KCNH3ALDH1A1MEN1KMT2AMAPT
SCHEMBL1924396 0.75 KCNH3 (0.83) KCNH3ALDH1A1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1479397-B1 2,4,6-TRIAMINO-1,3,5-TRIAZINE DERIVATIVE ASTELLAS PHARMA INC (JP) 2011-06-08 EP claimed
US-7375222-B2 2,4,6-Triamino-1,3,5-triazine derivative ASTELLAS PHARMA INC. (JP) 2008-05-20 US claimed
US-20120088772-A1 NOVEL PHARMACEUTICAL COMPOSITION FOR PREVENTION AND/OR TREATMENT OF ATTENTION DEFICIT/HYPERACTIVITY DISORDER ASTELLAS PHARMA INC. (JP) 2012-04-12 US disclosed
US-20100256152-A1 NOVEL PHARMACEUTICAL COMPOSITION FOR TREATMENT OF SCHIZOPHRENIA ASTELLAS PHARMA INC. (JP) 2010-10-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100256152-A1 NOVEL PHARMACEUTICAL COMPOSITION FOR TREATMENT OF SCHIZOPHRENIA KCNAB1, KCNN1, SCN1A KCNH3 81/4885ALDH1A1 3513/4885MEN1 3776/4885
US-20120088772-A1 NOVEL PHARMACEUTICAL COMPOSITION FOR PREVENTION AND/OR TREATMENT OF ATTENTION DEFICIT/HYPERACTIVITY DISORDER SLC6A3, ATP1A2, SLC6A1 KCNH3 105/4885ALDH1A1 722/4885MEN1 4082/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.