SCHEMBL1924841

SCHEMBL1924841

Cc1ccc2c(=O)c(-c3ccccc3)cn(CC(=O)N3CC(C)CC(C)C3)c2c1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
KDM4E B2RXH2 2/20 0.43
RECQL P46063 1/20 0.43
USP10 Q14694 2/20 0.42
GRIN2B Q13224 7/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1923600 0.89 SMN1; SMN2 (0.46) ALDH1A1SMN1; SMN2KMT2AKDM4EUSP10
SCHEMBL1923991 0.89 ALDH1A1 (0.47) ALDH1A1SMN1; SMN2MEN1KMT2AKDM4E
SCHEMBL1923580 0.85 MAPT (0.50) ALDH1A1USP10GRIN2B
SCHEMBL1923726 0.85 MAPT (0.51) ALDH1A1USP10GRIN2B
SCHEMBL1923633 0.84 USP10 (0.46) ALDH1A1MEN1KMT2AUSP10GRIN2B
SCHEMBL1923398 0.84 USP10 (0.49) ALDH1A1USP10GRIN2B
SCHEMBL1923300 0.84 USP10 (0.49) ALDH1A1SMN1; SMN2KMT2AUSP10GRIN2B
SCHEMBL1923418 0.83 ATM (0.51) ALDH1A1SMN1; SMN2MEN1KMT2AUSP10
SCHEMBL1923720 0.82 USP10 (0.40) ALDH1A1SMN1; SMN2USP10GRIN2B
SCHEMBL1924088 0.81 PTGDR2 (0.47) ALDH1A1KMT2AKDM4EUSP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2064185-B1 1H-QUINOLIN-4-ONE COMPOUNDS, WITH AFFINITY FOR THE GABA RECEPTOR, PROCESSES, USES AND COMPOSITIONS FERRER INT (ES) 2011-06-08 EP claimed
US-20100168099-A1 1H-QUINOLIN-4-ONE COMPOUNDS, WITH AFFINITY FOR THE GABA RECEPTOR, PROCESSES, USES AND COMPOSITIONS FERRER INTERNACIONAL, S.A. (ES) 2010-07-01 US claimed
EP-1886996-A1 1H-Quinolin-4-one compounds, with affinity for the GABA receptor, processes, uses and compositions FERRER INTERNACIONAL, S.A. (ES) 2008-02-13 EP claimed
EP-2064185-B1 1H-QUINOLIN-4-ONE COMPOUNDS, WITH AFFINITY FOR THE GABA RECEPTOR, PROCESSES, USES AND COMPOSITIONS FERRER INT (ES) 2011-06-08 EP disclosed
US-20100168099-A1 1H-QUINOLIN-4-ONE COMPOUNDS, WITH AFFINITY FOR THE GABA RECEPTOR, PROCESSES, USES AND COMPOSITIONS FERRER INTERNACIONAL, S.A. (ES) 2010-07-01 US disclosed
EP-1886996-A1 1H-Quinolin-4-one compounds, with affinity for the GABA receptor, processes, uses and compositions FERRER INTERNACIONAL, S.A. (ES) 2008-02-13 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100168099-A1 1H-QUINOLIN-4-ONE COMPOUNDS, WITH AFFINITY FOR THE GABA RECEPTOR, PROCESSES, USES AND COMPOSITIONS GABRA1, GABRA4, GABRA2 ALDH1A1 722/4885SMN1; SMN2 1630/4885MEN1 3307/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.