SCHEMBL19249082

SCHEMBL19249082

O=C(O)c1ccc(COc2cc(Br)cc3[nH]ncc23)cc1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RXRA P19793 9/20 0.48
RXRB P28702 8/20 0.48
FOLH1 Q04609 1/20 0.46
IDO1 P14902 3/20 0.46
TDO2 P48775 2/20 0.46
MRGPRX4 Q96LA9 1/20 0.44
HPGD P15428 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
RXRG P48443 6/20 0.43
CYP4F2 P78329 1/20 0.43
CYP4A11 Q02928 1/20 0.43
XDH P47989 1/20 0.43
MAP4K4 O95819 1/20 0.42
PIM1 P11309 1/20 0.41
PIM2 Q9P1W9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19248989 0.87 MRGPRX4 (0.53) FOLH1IDO1TDO2MRGPRX4HPGD
SCHEMBL19249081 0.87 MAPT (0.46) IDO1TDO2NPC1RAB9ASMN1; SMN2
SCHEMBL17440928 0.81 MAOB (0.45) IDO1TDO2NPC1RAB9ASMN1; SMN2
SCHEMBL19248986 0.78 CCR5 (0.48) IDO1TDO2MRGPRX4NPC1RAB9A
SCHEMBL19249343 0.76 TDO2 (0.74) IDO1TDO2
SCHEMBL17440906 0.72 IDO1 (0.51) IDO1TDO2
SCHEMBL19248997 0.72 NPC1 (0.52) IDO1TDO2HPGDNPC1RAB9A
SCHEMBL29151981 0.71 RXRA (0.49) RXRARXRBFOLH1MRGPRX4HPGD
SCHEMBL30631225 0.71 RXRA (0.49) RXRARXRBFOLH1MRGPRX4HPGD
SCHEMBL19249080 0.71 IDO1 (0.51) IDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017133258-A1 1H-INDAZOLE DERIVATIVE AND USE THEREOF AS IDO INHIBITOR 西华大学 2017-08-10 WO disclosed