SCHEMBL19251157

SCHEMBL19251157

CC1(C)COB(c2cccnc2N)O1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
MEN1 O00255 1/20 0.30
LMNA P02545 1/20 0.30
HSP90AA1 P07900 1/20 0.30
HSP90AB1 P08238 1/20 0.30
MAPT P10636 1/20 0.30
HTT P42858 1/20 0.30
BLM P54132 1/20 0.30
KMT2A Q03164 1/20 0.30
HIF1A Q16665 1/20 0.30
NAPRT Q6XQN6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19661719 0.82 LMNA (0.30) LMNA
SCHEMBL29468995 0.79 NOS3 (0.42) NOS3NOS1NOS2MEN1LMNA
SCHEMBL1114298 0.79 NOS3 (0.42) NOS3NOS1NOS2MEN1LMNA
SCHEMBL28402709 0.78 PLCG1 (0.32)
SCHEMBL24422669 0.74 CYP3A4 (0.39)
SCHEMBL28546786 0.72 TSHR (0.31)
SCHEMBL22570988 0.72 NOS3 (0.36) NOS3NOS1NOS2
SCHEMBL29592069 0.71 TAAR1 (0.33) LMNA
SCHEMBL29592082 0.71 ALDH1A1 (0.30)
SCHEMBL21003778 0.70 CYP2A6 (0.32) MAPTNAPRT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9732083-B2 Tricyclic gyrase inhibitors MERCK SHARP & DOHME CORP. (US) 2017-08-15 US disclosed