SCHEMBL24422669

SCHEMBL24422669

Cc1c(N)cccc1B1OCC(C)(C)O1

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.39
TSHR P16473 1/20 0.39
PIK3CA P42336 1/20 0.39
ALDH1A1 P00352 1/20 0.38
CD44 P16070 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1066081 0.84 CYP3A4 (0.42) CYP3A4TSHRPIK3CAALDH1A1CD44
SCHEMBL28589703 0.81 JAK2 (0.38) ALDH1A1
SCHEMBL29503402 0.78 CYP3A4 (0.46) CYP3A4TSHRPIK3CAALDH1A1CD44
SCHEMBL106726 0.78 CYP3A4 (0.46) CYP3A4TSHRPIK3CAALDH1A1CD44
SCHEMBL28546786 0.77 TSHR (0.31) TSHR
SCHEMBL30849833 0.75
SCHEMBL19251157 0.74 NOS3 (0.37)
SCHEMBL20805277 0.74 BACE1 (0.30)
SCHEMBL28499705 0.73 ALDH1A1 (0.37) TSHRALDH1A1
SCHEMBL29592069 0.72 TAAR1 (0.33) CYP3A4TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022099018-A1 PROCESS OF PREPARING A PD-1/PD-L1 INHIBITOR INCYTE CORPORATION (US) 2022-05-12 WO disclosed