SCHEMBL19251203

SCHEMBL19251203

CC(C)(S)OCc1ccnc(N)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 5/20 0.53
NOS2 P35228 5/20 0.53
NOS1 P29475 4/20 0.53
GABRP O00591 2/20 0.44
GABRD O14764 2/20 0.44
GABRA1 P14867 2/20 0.44
GABRB1 P18505 2/20 0.44
GABRG2 P18507 2/20 0.44
GABRB3 P28472 2/20 0.44
GABRA5 P31644 2/20 0.44
GABRA3 P34903 2/20 0.44
GABRA2 P47869 2/20 0.44
GABRB2 P47870 2/20 0.44
GABRA4 P48169 2/20 0.44
GABRE P78334 2/20 0.44
GABRA6 Q16445 2/20 0.44
GABRG1 Q8N1C3 2/20 0.44
GABRG3 Q99928 2/20 0.44
GABRQ Q9UN88 2/20 0.44
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20288434 0.86 NOS3 (0.56) NOS3NOS2NOS1GABRPGABRD
SCHEMBL19251204 0.82 NOS3 (0.56) NOS3NOS2NOS1GABRPGABRD
SCHEMBL19251202 0.79 LOXL2 (0.56) LOXLOXL2NUDT1AAK1NPC1
SCHEMBL2118728 0.78 NOS3 (0.64) NOS3NOS2NOS1GABRPGABRD
SCHEMBL29883563 0.78 NOS3 (0.64) NOS3NOS2NOS1GABRPGABRD
SCHEMBL331281 0.75 NOS3 (0.51) NOS3NOS2NOS1GABRPGABRD
SCHEMBL26799850 0.74 LOXL2 (0.38) LOXL2RAB9A
SCHEMBL16316855 0.74 NOS3 (0.63) NOS3NOS2NOS1GABRPGABRD
SCHEMBL10087561 0.73 NOS3 (0.62) NOS3NOS2NOS1GABRPGABRD
SCHEMBL13302576 0.72 NOS3 (0.56) NOS3NOS2NOS1GABRPGABRD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9878987-B2 HSP70 modulators and methods for making and using the same MEMORIAL SLOAN KETTERING CANCER CENTER (US) 2018-01-30 US disclosed
US-20170233352-A1 HSP70 MODULATORS AND METHODS FOR MAKING AND USING THE SAME MEMORIAL SLOAN KETTERING CANCER CENTER 2017-08-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170233352-A1 HSP70 MODULATORS AND METHODS FOR MAKING AND USING THE SAME HSPA2, HSP90AA1, HSP90AB1 NOS3 3133/4885NOS2 1682/4885NOS1 2664/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.