SCHEMBL19254586

SCHEMBL19254586

CCOc1ccc(-c2nc(C#N)c3[nH]c(=O)n(CC)c3n2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 3/20 0.41
NSD2 O96028 1/20 0.41
NSD3 Q9BZ95 1/20 0.41
KDM4E B2RXH2 6/20 0.40
ALDH1A1 P00352 5/20 0.40
CTSS P25774 2/20 0.40
CTSK P43235 2/20 0.40
HPGD P15428 3/20 0.39
MAPK1 P28482 3/20 0.39
HSD17B10 Q99714 3/20 0.39
MAPT P10636 2/20 0.39
LMNA P02545 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
RECQL P46063 1/20 0.39
TP53 P04637 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ADORA1 P30542 2/20 0.38
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19254587 0.88 ALDH1A1 (0.41) ADORA2BKDM4EALDH1A1CTSSCTSK
SCHEMBL19207635 0.80 HDAC3 (0.60) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL19207629 0.79 MEN1 (0.47) KDM4EALDH1A1HPGDHSD17B10MAPT
SCHEMBL19207423 0.79 CSNK2A1 (0.49) ADORA2BKDM4EALDH1A1HPGDHSD17B10
SCHEMBL19254333 0.76 CSNK2A1 (0.47) KDM4EALDH1A1HPGDMAPK1HSD17B10
SCHEMBL19207433 0.76 CSNK2A1 (0.41) KDM4EMAPK1HSD17B10MAPTLMNA
SCHEMBL19207434 0.76 CSNK2A1 (0.47) KDM4EALDH1A1HPGDMAPK1HSD17B10
SCHEMBL19207491 0.69 CSNK2A1 (0.49) ADORA2BKDM4EALDH1A1HPGDHSD17B10
SCHEMBL19207408 0.68 THRB (0.49) KDM4EALDH1A1HPGDMAPTLMNA
SCHEMBL19254750 0.67 CSNK2A1 (0.55) KDM4EALDH1A1HPGDMAPK1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017136689-A1 PURINE COMPOUNDS POSSESSING ANTICANCER ACTIVITY ACADEMIA SINICA (TW) 2017-08-10 WO disclosed