SCHEMBL19256724

SCHEMBL19256724

Cn1nnn(-c2cc([N+](=O)[O-])c(F)cc2[C@H]2CC2C(F)(F)F)c1=O

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.32
GAA P10253 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30
MAPT P10636 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1936956 1.00 ALDH1A1 (0.32) ALDH1A1GAACYP1A2CYP2D6MAPT
SCHEMBL9886504 1.00 ALDH1A1 (0.32) ALDH1A1GAACYP1A2CYP2D6MAPT
SCHEMBL1945616 0.83 ALDH1A1 (0.37) ALDH1A1GAACYP1A2CYP2D6MAPT
SCHEMBL1943801 0.82 DPP4 (0.30)
SCHEMBL1943802 0.82 DPP4 (0.30)
SCHEMBL9886503 0.82 DPP4 (0.30)
SCHEMBL12539977 0.76 ALDH1A1 (0.35) ALDH1A1GAAMAPT
SCHEMBL10199255 0.76 LMNA (0.42) ALDH1A1MAPT
SCHEMBL1944352 0.76 MAPT (0.40) ALDH1A1GAACYP1A2CYP2D6MAPT
SCHEMBL1942929 0.76 PKM (0.35) ALDH1A1CYP1A2CYP2D6MAPTCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9732070-B2 Protein kinase C inhibitors and uses thereof RIGEL PHARMACEUTICALS, INC. (US) 2017-08-15 US disclosed