SCHEMBL19259529

SCHEMBL19259529

c1cc2[nH]cc3ccccc3c-2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.47
ALPL P05186 1/20 0.47
GAA P10253 1/20 0.47
MCL1 Q07820 1/20 0.41
GSK3B P49841 1/20 0.41
CDK5 Q00535 1/20 0.41
CDK5R1 Q15078 1/20 0.41
NISCH Q9Y2I1 1/20 0.38
ALDH1A1 P00352 4/20 0.36
HSD17B10 Q99714 4/20 0.36
TSHR P16473 3/20 0.36
MAPK1 P28482 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
HPGD P15428 2/20 0.36
CASP1 P29466 1/20 0.36
HIF1A Q16665 1/20 0.36
ATM Q13315 1/20 0.36
IKBKE Q14164 1/20 0.36
TBK1 Q9UHD2 1/20 0.36
PTPN1 P18031 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2289477 0.81 KDM4E (0.50) KDM4EALPLGAAMCL1GSK3B
SCHEMBL5133946 0.75 KDM4E (0.45) KDM4EALPLGAAMCL1GSK3B
SCHEMBL2046783 0.74 MAPK1 (0.32) KDM4EALDH1A1HSD17B10TSHRMAPK1
SCHEMBL5576841 0.74 PRKCZ (0.43) IKBKETBK1CYP1A2
SCHEMBL28065244 0.72 HPRT1 (0.52) KDM4EALPLGAAGSK3BCDK5
SCHEMBL378547 0.72 DNMT1 (0.38) KDM4EALPLGAAMCL1ALDH1A1
SCHEMBL26259996 0.72 AURKA (0.48) KDM4EALPLGAAGSK3BCDK5
Hydrochloric Acid SCHEMBL6554454 0.71 DNMT1 (0.37) KDM4EALPLGAAMCL1ALDH1A1
SCHEMBL27263879 0.71 ALDH1A1 (0.53) KDM4EALPLGAAGSK3BNISCH
SCHEMBL25302086 0.70 ALDH1A1 (0.59) KDM4EALPLGAANISCHALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3416946-A1 TETRACYCLIC PYRIDONE COMPOUNDS AS ANTIVIRALS Novartis AG (CH) 2018-12-26 EP disclosed
WO-2017140821-A1 TETRACYCLIC PYRIDONE COMPOUNDS AS ANTIVIRALS NOVARTIS AG (CH) 2017-08-24 WO disclosed