SCHEMBL19265367

SCHEMBL19265367

Cc1cc(Cl)cc(C(C)(C)C(F)(F)F)c1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RAPGEF4 Q8WZA2 3/20 0.41
PGK1 P00558 1/20 0.34
PGK2 P07205 1/20 0.34
PDE2A O00408 1/20 0.33
NR3C1 P04150 1/20 0.32
NR3C2 P08235 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25767125 0.84 PGK1 (0.40) RAPGEF4PGK1PGK2PDE2A
SCHEMBL22808889 0.83 RAPGEF4 (0.43) RAPGEF4PGK1PGK2NR3C1NR3C2
SCHEMBL902818 0.80 RAPGEF4 (0.58) RAPGEF4PGK1PGK2
SCHEMBL16261286 0.78 GABRA1 (0.41) RAPGEF4PGK1PGK2PDE2A
SCHEMBL8826911 0.78 POLB (0.41) RAPGEF4
SCHEMBL15459372 0.78 PDE2A (0.32) RAPGEF4PDE2A
SCHEMBL24355332 0.76 RAPGEF4 (0.39) RAPGEF4PGK1PGK2NR3C1NR3C2
SCHEMBL16579376 0.74 RAPGEF4 (0.40) RAPGEF4PDE2A
SCHEMBL19507024 0.74 MEN1 (0.38) RAPGEF4PGK1PGK2NR3C1NR3C2
SCHEMBL22783306 0.73 RAPGEF4 (0.40) RAPGEF4PGK1PGK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2875021-B1 BETA AMINO ACID DERIVATIVES AS INTEGRIN ANTAGONISTS UNIV SAINT LOUIS (US) 2017-08-23 EP disclosed