SCHEMBL19275201

SCHEMBL19275201

O=C(CI)N1CCN(CC2CCOCC2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 1/20 0.49
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HRH3 Q9Y5N1 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CACNA2D1 P54289 2/20 0.39
CACNA1B Q00975 2/20 0.39
CACNB1 Q02641 2/20 0.39
CACNA1C Q13936 1/20 0.39
THRB P10828 1/20 0.39
KDM4E B2RXH2 4/20 0.38
LMNA P02545 1/20 0.38
RAB9A P51151 1/20 0.38
GBA1 P04062 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
ALDH1A1 P00352 4/20 0.37
NAMPT P43490 2/20 0.37
TDP1 Q9NUW8 1/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18909105 0.84 TACR2 (0.49) TACR2ALOX15TSHRHSD17B10HRH3
SCHEMBL3602019 0.81 TACR2 (0.49) TACR2ALOX15TSHRHSD17B10HRH3
SCHEMBL22030492 0.80 TACR2 (0.46) TACR2ALOX15TSHRHSD17B10HRH3
SCHEMBL24585267 0.79 TACR2 (0.46) TACR2ALOX15TSHRHSD17B10HRH3
SCHEMBL2262931 0.76 L3MBTL1 (0.61) ALOX15TSHRHSD17B10L3MBTL1LMNA
SCHEMBL18909453 0.74 ALOX15 (0.55) ALOX15TSHRHSD17B10L3MBTL1CACNA2D1
SCHEMBL26065145 0.73 USP2 (0.58) L3MBTL1KDM4ELMNARAB9AALDH1A1
SCHEMBL9275712 0.72 ALDH1A1 (0.48) ALOX15TSHRHSD17B10L3MBTL1KDM4E
SCHEMBL19275281 0.71 THRB (0.50) TACR2ALOX15TSHRHSD17B10L3MBTL1
SCHEMBL18909230 0.71 THRB (0.53) ALOX15TSHRHSD17B10THRBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017140825-A1 THERAPEUTIC COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2017-08-24 WO disclosed