SCHEMBL19288503

SCHEMBL19288503

CN1CN(C)C(=O)c2c(I)cccc2C1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.37
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
USP2 O75604 1/20 0.35
CASP1 P29466 1/20 0.35
BRCA1 P38398 1/20 0.35
CASP7 P55210 1/20 0.35
CES1 P23141 2/20 0.34
BCHE P06276 1/20 0.34
TDP2 O95551 1/20 0.34
DPP4 P27487 1/20 0.33
ALDH1A1 P00352 3/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 2/20 0.32
HPGD P15428 2/20 0.32
KDM4E B2RXH2 1/20 0.32
GAA P10253 1/20 0.32
CASP3 P42574 1/20 0.32
HTR2B P41595 1/20 0.32
TMEM97 Q5BJF2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15219284 0.80 DPP4 (0.47) MEN1KMT2ADPP4ALDH1A1POLB
SCHEMBL4369262 0.79 MEN1 (0.53) MEN1KMT2AUSP2CASP1BRCA1
SCHEMBL30725967 0.79 MEN1 (0.53) MEN1KMT2AUSP2CASP1BRCA1
SCHEMBL11916140 0.76 CA2 (0.34) PARP1MEN1KMT2AUSP2CASP1
SCHEMBL25767173 0.73 PARP1 (0.57) PARP1KMT2ATDP2
SCHEMBL25772610 0.73 POLB (0.37) PARP1MEN1KMT2AALDH1A1POLB
SCHEMBL11093043 0.72 HSPA1A (0.33) MEN1KMT2AUSP2CASP1BRCA1
SCHEMBL24265738 0.70 POLB (0.50) MEN1KMT2AALDH1A1POLB
SCHEMBL6362382 0.69 CES1 (0.48) CES1BCHEALDH1A1MAPTHPGD
SCHEMBL11068602 0.69 ALDH1A1 (0.54) MEN1KMT2AUSP2CES1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3210609-A1 PHOSPHOROUS DERIVATIVES AS KINASE INHIBITORS ARIAD PHARMACEUTICALS, INC. (US) 2017-08-30 EP disclosed