SCHEMBL19306397

SCHEMBL19306397

O=C1CSC(c2ccc(F)cc2)N1Cc1ccccc1

nearest known ligand 0.78

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.78
MEN1 O00255 5/20 0.78
MAPT P10636 1/20 0.74
POLB P06746 2/20 0.69
CYP2C9 P11712 1/20 0.69
CYP2C19 P33261 1/20 0.69
HPGD P15428 3/20 0.63
LMNA P02545 3/20 0.63
SMN1; SMN2 Q16637 2/20 0.63
L3MBTL1 Q9Y468 2/20 0.63
ALOX12 P18054 1/20 0.63
NPSR1 Q6W5P4 1/20 0.63
GAA P10253 2/20 0.62
HTT P42858 1/20 0.62
ATM Q13315 1/20 0.61
ALDH1A1 P00352 3/20 0.58
KDM4E B2RXH2 1/20 0.57
PSMD14 O00487 1/20 0.55
GPR55 Q9Y2T6 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19306513 0.87 MEN1 (0.71) KMT2AMEN1MAPTCYP2C9CYP2C19
SCHEMBL5152843 0.84 MEN1 (0.75) KMT2AMEN1MAPTPOLBCYP2C9
SCHEMBL5152438 0.82 MEN1 (0.72) KMT2AMEN1MAPTPOLBCYP2C9
SCHEMBL5151573 0.82 MAPT (0.67) KMT2AMEN1MAPTPOLBCYP2C9
SCHEMBL5155057 0.82 KMT2A (0.67) KMT2AMEN1MAPTPOLBCYP2C9
SCHEMBL28630573 0.81 MEN1 (0.57) KMT2AMEN1MAPTPOLBCYP2C9
SCHEMBL19305954 0.80 MEN1 (0.81) KMT2AMEN1MAPTPOLBCYP2C9
SCHEMBL5156737 0.80 KMT2A (0.61) KMT2AMEN1MAPTPOLBCYP2C9
SCHEMBL5151457 0.78 MEN1 (0.63) KMT2AMEN1MAPTALDH1A1
SCHEMBL6919581 0.78 MEN1 (0.65) KMT2AMEN1MAPTPOLBCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3426246-B1 THIAZOLIDINONE COMPOUNDS AND USE THEREOF NATIONAL HEALTH RES INST (TW) 2024-05-01 EP disclosed
CN-108883099-B Thiazolidinone compounds and use thereof 石全 2021-09-28 CN disclosed
US-10544113-B2 Thiazolidinone compounds and use thereof NATIONAL HEALTH RESEARCH INSTITUTE (TW) 2020-01-28 US disclosed
US-10544113-B2 Thiazolidinone compounds and use thereof NATIONAL HEALTH RESEARCH INSTITUTE (TW) 2020-01-28 US disclosed
EP-3426246-A1 THIAZOLIDINONE COMPOUNDS AND USE THEREOF National Health Research Institutes (TW) 2019-01-16 EP disclosed
CN-108883099-A THIAZOLIDINONE COMPOUNDS AND USE THEREOF 石全 2018-11-23 CN disclosed
WO-2017155910-A1 THIAZOLIDINONE COMPOUNDS AND USE THEREOF NATIONAL HEALTH RESEARCH INSTITUTES (TW) 2017-09-14 WO disclosed
WO-2017155910-A1 THIAZOLIDINONE COMPOUNDS AND USE THEREOF NATIONAL HEALTH RESEARCH INSTITUTES (TW) 2017-09-14 WO disclosed
US-20170253569-A1 THIAZOLIDINONE COMPOUNDS AND USE THEREOF REGENTS OF THE UNIVERSITY OF MINNESOTA 2017-09-07 US disclosed
US-20170253569-A1 THIAZOLIDINONE COMPOUNDS AND USE THEREOF REGENTS OF THE UNIVERSITY OF MINNESOTA 2017-09-07 US disclosed
US-20170253569-A1 THIAZOLIDINONE COMPOUNDS AND USE THEREOF REGENTS OF THE UNIVERSITY OF MINNESOTA 2017-09-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10544113-B2 Thiazolidinone compounds and use thereof OPRL1, OPRD1, OPRK1 KMT2A 3536/4885MEN1 4566/4885MAPT 1648/4885
US-20170253569-A1 THIAZOLIDINONE COMPOUNDS AND USE THEREOF OPRL1, OPRD1, OPRK1 KMT2A 3536/4885MEN1 4566/4885MAPT 1648/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.