SCHEMBL19308451

SCHEMBL19308451

CC(=O)CC(=O)Nc1ccc2[nH]c3ccccc3c2c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.74
KMT2A Q03164 2/20 0.74
MTNR1A P48039 2/20 0.74
MTNR1B P49286 2/20 0.74
P2RY12 Q9H244 2/20 0.63
NPY5R Q15761 1/20 0.60
PARP1 P09874 3/20 0.56
TNKS O95271 1/20 0.56
PARP15 Q460N3 1/20 0.56
PARP14 Q460N5 1/20 0.56
PARP10 Q53GL7 1/20 0.56
PARP12 Q9H0J9 1/20 0.56
TNKS2 Q9H2K2 1/20 0.56
PARP2 Q9UGN5 1/20 0.56
PARP4 Q9UKK3 1/20 0.56
PARP3 Q9Y6F1 1/20 0.56
MEN1 O00255 1/20 0.56
ALDH1A1 P00352 1/20 0.56
CYP1A2 P05177 1/20 0.56
CYP2C19 P33261 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19308466 0.86 P2RY12 (0.71) KDM4EKMT2AMTNR1AMTNR1BP2RY12
SCHEMBL31488126 0.85 MTNR1A (1.00) KDM4EKMT2AMTNR1AMTNR1BP2RY12
SCHEMBL7722965 0.85 MTNR1A (1.00) KDM4EKMT2AMTNR1AMTNR1BP2RY12
SCHEMBL4728869 0.83 PARP1 (0.79) KDM4EKMT2AMTNR1AMTNR1BP2RY12
SCHEMBL4728731 0.82 CCKBR (0.65) KDM4EKMT2AMTNR1AMTNR1BP2RY12
SCHEMBL4726206 0.82 P2RY12 (0.73) KDM4EKMT2AMTNR1AMTNR1BP2RY12
SCHEMBL4726214 0.82 P2RY12 (0.73) KDM4EKMT2AMTNR1AMTNR1BP2RY12
SCHEMBL21855490 0.80 KDM4E (0.74) KDM4EKMT2AMTNR1AMTNR1BP2RY12
SCHEMBL30227292 0.80 KDM4E (0.74) KDM4EKMT2AMTNR1AMTNR1BP2RY12
SCHEMBL19308465 0.80 P2RY12 (0.73) KDM4EKMT2AMTNR1AMTNR1BP2RY12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9751851-B2 Molecules and compositions that inhibit gram negative bacteria and their uses THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2017-09-05 US disclosed