SCHEMBL19334382

SCHEMBL19334382

Cn1c(COc2ccc([N+](=O)O)cc2)nnc1SCC(=O)O

nearest known ligand 0.67

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.67
ALDH1A1 P00352 4/20 0.67
NPC1 O15118 1/20 0.66
KDM4E B2RXH2 3/20 0.64
MEN1 O00255 2/20 0.57
GAA P10253 2/20 0.57
MAPT P10636 2/20 0.56
HPGD P15428 1/20 0.56
CRHBP P24387 1/20 0.56
CRHR2 Q13324 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
HSD17B10 Q99714 1/20 0.55
PKM P14618 2/20 0.54
POLB P06746 1/20 0.54
TSHR P16473 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.53
HTT P42858 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13401700 0.90 ALDH1A1 (0.82) KMT2AALDH1A1NPC1KDM4EMEN1
SCHEMBL4204174 0.74 ALDH1A1 (0.72) KMT2AALDH1A1NPC1MEN1GAA
SCHEMBL4214358 0.74 LMNA (0.71) KMT2AALDH1A1NPC1MEN1GAA
SCHEMBL11887417 0.70 KMT2A (0.80) KMT2AALDH1A1NPC1MEN1MAPT
SCHEMBL6405241 0.68 L3MBTL1 (0.84) KMT2AALDH1A1MEN1MAPTHPGD
SCHEMBL6404334 0.68 GAA (0.71) KMT2AALDH1A1NPC1KDM4EMEN1
SCHEMBL6407491 0.68 PKM (0.60) KMT2AALDH1A1NPC1KDM4EGAA
SCHEMBL6405274 0.67 GAA (0.74) KMT2AALDH1A1NPC1MEN1GAA
SCHEMBL6412252 0.65 PKM (0.56) KMT2AALDH1A1KDM4EMEN1GAA
SCHEMBL5968206 0.65 ALDH1A1 (0.54) KMT2AALDH1A1NPC1MEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9757375-B2 Compounds that inhibit human DNA ligases and methods of treating cancer UNIVERSITY OF MARYLAND, BALTIMORE (US) 2017-09-12 US disclosed