SCHEMBL1933748

SCHEMBL1933748

O=C(O)c1cc(F)cc(B(O)O)c1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 1/20 0.55
HCAR2 Q8TDS4 1/20 0.48
CES2 O00748 2/20 0.43
CES1 P23141 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.41
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
BCL2L1 Q07817 1/20 0.38
BAD Q92934 1/20 0.38
TTR P02766 1/20 0.38
PPARA Q07869 1/20 0.37
TPMT P51580 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30506535 1.00 HCAR1 (0.55) HCAR1HCAR2CES2CES1L3MBTL1
SCHEMBL22400317 0.93 HCAR1 (0.48) HCAR1HCAR2CES2CES1L3MBTL1
SCHEMBL918608 0.84 CA12 (0.46) CA12CA1CA2CA7CA9
SCHEMBL6733033 0.84 CA1 (0.46) HCAR1CA12CA1CA2CA7
SCHEMBL5151998 0.82 CES2 (0.41) HCAR1HCAR2CES2CES1
SCHEMBL29821986 0.82 PARP1 (0.52) HCAR1HCAR2CES2CES1
SCHEMBL14120715 0.82 PARP1 (0.52) HCAR1HCAR2CES2CES1
SCHEMBL28959114 0.80 APP (0.46) HCAR1PPARA
SCHEMBL157714 0.79 HCAR1 (0.73) HCAR1HCAR2CES2CES1L3MBTL1
SCHEMBL336433 0.79 HCAR1 (0.73) HCAR1HCAR2CES2CES1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 59 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111146496-B Polymer electrolyte and lithium ion battery containing same 珠海冠宇电池股份有限公司 2021-07-13 CN claimed
CN-112679535-A Small molecule PAD4 inhibitor and preparation method and application thereof 首都医科大学 2021-04-20 CN claimed
CN-111162313-A Polymer electrolyte and lithium ion battery 珠海冠宇电池有限公司 2020-05-15 CN claimed
CN-111146496-A Polymer electrolyte and lithium ion battery containing same 珠海冠宇电池有限公司 2020-05-12 CN claimed
US-12637436-B2 Metabotropic glutamate receptor negative allosteric modulators (NAMs) and uses thereof Sanford Burnham Prebys Medical Discovery Institute (US) 2026-05-26 US disclosed
EP-4323354-B1 2-((4-((S)-2-(4-CHLORO-2-FLUOROPHENYL)-2-METHYLBENZO[D][1,3]DIOXOL-4-YL)PIPERIDIN-1-YL)METHYL)-1-(((S)-OXETAN-2-YL)METHYL)-1H-IMIDAZOLE DERIVATIVES AS ACTIVATORS OF THE GLP1 RECEPTOR FOR THE TREATMENT OF OBESITY NOVARTIS AG (CH) 2025-12-17 EP disclosed
US-20250179000-A1 METABOTROPIC GLUTAMATE RECEPTOR POSITIVE ALLOSTERIC MODULATORS (PAMS) AND USES THEREOF Sanford Burnham Prebys Medical Discovery Institute 2025-06-05 US disclosed
CN-120058751-A Pleuromutilin derivative with arylboronic acid or arylboronic acid ester fragment, and preparation method and application thereof 中国医学科学院药物研究所 2025-05-30 CN disclosed
CN-119192845-B Preparation method of high-temperature-resistant high-heat-conductivity PPS composite material 东莞市普万光电散热科技有限公司 2025-03-14 CN disclosed
CN-118772595-B Wear-resistant glass fiber reinforced plastic well lid containing polyester and preparation method thereof 山东金光复合材料股份有限公司 2025-01-24 CN disclosed
CN-118772595-A Wear-resistant glass fiber reinforced plastic well lid containing polyester and preparation method thereof 山东金光复合材料股份有限公司 2024-10-15 CN disclosed
US-20240182456-A1 2-((4-((S)-2-(4-CHLORO-2-FLUOROPHENYL)-2-METHYLBENZO[D][1,3]DIOXOL-4-YL)PIPERIDIN-1-YL)METHYL)-1-(((S)-OXETAN-2-YL)METHYL)-1H-IMIDAZOLE DERIVATIVES AS ACTIVATORS OF THE GLP1 RECEPTOR FOR THE TREATMENT OF OBESITY NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC. 2024-06-06 US disclosed
US-20150119390-A1 IMIDAZOTHIADIAZOLE AND IMIDAZOPYRIDAZINE DERIVATIVES AS PROTEASE ACTIVATED RECEPTOR 4 (PAR4) INHIBITORS FOR TREATING PLATELET AGGREGATION BRISTOL-MYERS SQUIBB COMPANY 2015-04-30 US disclosed
EP-2855489-A1 IMIDAZOTHIADIAZOLE AND IMIDAZOPYRIDAZINE DERIVATIVES AS PROTEASE ACTIVATED RECEPTOR 4 (PAR4) INHIBITORS FOR TREATING PLATELET AGGREGATION Bristol-Myers Squibb Company (US) 2015-04-08 EP disclosed
EP-2507236-B1 Triazolopyridine derivates BAYER IP GMBH (DE) 2014-12-17 EP disclosed
WO-2014159559-A1 FUSED FURANS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2014-10-02 WO disclosed
WO-2014159559-A1 FUSED FURANS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2014-10-02 WO disclosed
WO-2013163241-A1 IMIDAZOTHIADIAZOLE AND IMIDAZOPYRIDAZINE DERIVATIVES AS PROTEASE ACTIVATED RECEPTOR 4 (PAR4) INHIBITORS FOR TREATING PLATELET AGGREGATION BRISTOL-MYERS SQUIBB COMPANY (US) 2013-10-31 WO disclosed
EP-2507236-A1 TRIAZOLOPYRIDINE DERIVATIVES Bayer Intellectual Property GmbH (DE) 2012-10-10 EP disclosed
WO-2011064328-A1 TRIAZOLOPYRIDINE DERIVATIVES BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2011-06-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250179000-A1 METABOTROPIC GLUTAMATE RECEPTOR POSITIVE ALLOSTERIC MODULATORS (PAMS) AND USES THEREOF GRM3, GRM2, GRM1 HCAR1 137/4885HCAR2 96/4885CES2 2588/4885
US-20240182456-A1 2-((4-((S)-2-(4-CHLORO-2-FLUOROPHENYL)-2-METHYLBENZO[D][1,3]DIOXOL-4-YL)PIPERIDIN-1-YL)METHYL)-1-(((S)-OXETAN-2-YL)METHYL)-1H-IMIDAZOLE DERIVATIVES AS ACTIVATORS OF THE GLP1 RECEPTOR FOR THE TREATMENT OF OBESITY GLP1R, GPR119, IRS1 HCAR1 964/4885HCAR2 627/4885CES2 1090/4885
US-20150119390-A1 IMIDAZOTHIADIAZOLE AND IMIDAZOPYRIDAZINE DERIVATIVES AS PROTEASE ACTIVATED RECEPTOR 4 (PAR4) INHIBITORS FOR TREATING PLATELET AGGREGATION F2RL3, F2R, F2RL1 HCAR1 351/4885HCAR2 495/4885CES2 2777/4885
US-12637436-B2 Metabotropic glutamate receptor negative allosteric modulators (NAMs) and uses thereof GRM3, GRM2, GRM1 HCAR1 338/4885HCAR2 167/4885CES2 1415/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.