SCHEMBL5151998

SCHEMBL5151998

CC(=O)c1cc(F)cc(B(O)O)c1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.41
CES1 P23141 3/20 0.41
CA5A P35218 1/20 0.40
HCAR1 Q9BXC0 1/20 0.35
HCAR2 Q8TDS4 1/20 0.34
PARP1 P09874 1/20 0.34
LMNA P02545 1/20 0.34
MAOB P27338 2/20 0.34
SLC6A3 Q01959 1/20 0.33
HDAC1 Q13547 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
ALDH1A1 P00352 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3785242 0.85 CA5A (0.48) CA5ALMNAKMT2A
SCHEMBL11303214 0.85 CA5A (0.48) CA5ALMNAKMT2A
SCHEMBL1933748 0.82 HCAR1 (0.55) CES2CES1HCAR1HCAR2
SCHEMBL30506535 0.82 HCAR1 (0.55) CES2CES1HCAR1HCAR2
SCHEMBL319123 0.80 CES2 (0.62) CES2CES1CA5AHCAR1HCAR2
SCHEMBL29821986 0.80 PARP1 (0.52) CES2CES1HCAR1HCAR2PARP1
SCHEMBL14120715 0.80 PARP1 (0.52) CES2CES1HCAR1HCAR2PARP1
SCHEMBL3764991 0.79 CES2 (0.38) CES2CES1HCAR1ALDH1A1KMT2A
SCHEMBL2013972 0.79 MAP4K4 (0.39) CES2CES1HDAC1HDAC6ALDH1A1
SCHEMBL29821598 0.79 CES2 (0.38) CES2CES1HCAR1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200361939-A1 MODULATORS OF ALPHA-1 ANTITRYPSIN VERTEX PHARMACEUTICALS INCORPORATED. 2020-11-19 US disclosed
US-20070060573-A1 Acyltryptophanols BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2007-03-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070060573-A1 Acyltryptophanols FSHR, NPY1R, NPY2R CES2 3951/4885CES1 2493/4885CA5A 3680/4885
US-20200361939-A1 MODULATORS OF ALPHA-1 ANTITRYPSIN SERPINA2, SERPINC1, SERPINA3 CES2 2440/4885CES1 166/4885CA5A 2689/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.