SCHEMBL1933757

SCHEMBL1933757

Cc1c[c]c2cccc(F)c2n1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.33
GAA P10253 3/20 0.33
LMNA P02545 2/20 0.33
RAB9A P51151 2/20 0.33
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
PRNP P04156 1/20 0.33
HPGD P15428 1/20 0.33
KMT2A Q03164 1/20 0.33
MAPT P10636 2/20 0.32
METAP2 P50579 1/20 0.32
CCR1 P32246 2/20 0.31
ACHE P22303 1/20 0.31
CCR5 P51681 1/20 0.31
MGAM O43451 1/20 0.31
SI P14410 1/20 0.31
MGAM2 Q2M2H8 1/20 0.31
AR P10275 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL315820 0.81 TP53 (0.37) SMN1; SMN2GAALMNARAB9AALDH1A1
SCHEMBL944682 0.79 ALDH1A1 (0.35) SMN1; SMN2GAALMNAALDH1A1MEN1
SCHEMBL27764064 0.77 NPC1 (0.36) SMN1; SMN2GAALMNARAB9AALDH1A1
SCHEMBL22093016 0.75 NQO2 (0.47) SMN1; SMN2GAALMNARAB9AALDH1A1
SCHEMBL5926098 0.70 PARP1 (0.37) SMN1; SMN2LMNARAB9AALDH1A1KDM4E
SCHEMBL378207 0.68 METAP2 (0.59) SMN1; SMN2LMNARAB9AMEN1KMT2A
SCHEMBL96433 0.68 CYP1A2 (0.45) SMN1; SMN2GAARAB9AALDH1A1KDM4E
SCHEMBL22126089 0.68 AR (0.37) SMN1; SMN2GAALMNARAB9AALDH1A1
SCHEMBL19189304 0.64 KDM4E (0.62) SMN1; SMN2GAALMNARAB9AALDH1A1
SCHEMBL1090860 0.63 KDM4E (0.35) GAAALDH1A1KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3682873-B1 SMAC MIMETICS FOR USE IN THE TREATMENT OF PERSISTENT HIV INFECTION WALTER & ELIZA HALL INST MEDICAL RES (AU) 2024-06-12 EP disclosed
US-11702401-B2 Compounds and methods of use MEDIVATION TECHNOLOGIES LLC (US) 2023-07-18 US disclosed
US-20220000847-A1 Compounds and Methods of Use MEDIVATION TECHNOLOGIES LLC (US) 2022-01-06 US disclosed
US-11053216-B2 Compounds and methods of use MEDIVATION TECHNOLOGIES LLC (US) 2021-07-06 US disclosed
CN-112957365-A Methods of treating intracellular infections 沃尔特和伊利莎豪医学研究所 2021-06-15 CN disclosed
CN-105451726-B Methods of treating intracellular infections 沃尔特和伊利莎豪医学研究所 2021-03-16 CN disclosed
EP-3013329-B1 SMAC MIMETICS FOR THE TREATMENT OF PERSISTENT INTRACELLULAR HBV INFECTION WALTER & ELIZA HALL INST MEDICAL RES (AU) 2020-08-05 EP disclosed
CN-111481669-A Methods of treating intracellular infections 沃尔特和伊利莎豪医学研究所 2020-08-04 CN disclosed
EP-3089971-B1 COMPOUNDS AND METHODS OF USE MEDIVATION TECH LLC (US) 2020-07-29 EP disclosed
EP-3682873-A1 SMAC MIMETICS FOR USE IN THE TREATMENT OF PERSISTENT HIV INFECTION The Walter and Eliza Hall Institute of Medical Research (AU) 2020-07-22 EP disclosed
WO-2015017520-A1 METHOD OF TREATMENT TETRALOGIC PHARMACEUTICALS CORP. (US) 2015-02-05 WO disclosed
WO-2014205516-A1 METHOD OF TREATING INTRACELLULAR INFECTION THE WALTER AND ELIZA HALL INSTITUTE OF MEDICAL RESEARCH (AU) 2014-12-31 WO disclosed
US-20140303090-A1 Smac Mimetic Therapy TETRALOGIC PHARMACEUTICALS CORPORATION (US) 2014-10-09 US disclosed
WO-2014022612-A1 COMBINATION THERAPY TETRALOGIC PHARMACEUTICALS CORPORATION (US) 2014-02-06 WO disclosed
US-20130196927-A1 Smac Mimetic Therapy TETRALOGIC PHARMACEUTICALS CORPORATION 2013-08-01 US disclosed
EP-2434889-A1 IAP INHIBITORS Tetralogic Pharmaceuticals Corp. (US) 2012-04-04 EP disclosed
EP-2434890-A1 IAP INHIBITORS Tetralogic Pharmaceuticals Corp. (US) 2012-04-04 EP disclosed
WO-2011068926-A1 IAP INHIBITORS TETRALOGIC PHARMACEUTICALS CORP. (US) 2011-06-09 WO disclosed
WO-2010138496-A1 IAP INHIBITORS TETRALOGIC PHARMACEUTICALS CORP. (US) 2010-12-02 WO disclosed
WO-2010138666-A1 IAP INHIBITORS TETRALOGIC PHARMACEUTICALS CORP. (US) 2010-12-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220000847-A1 Compounds and Methods of Use TGFB2, TGFB1, HDGF SMN1; SMN2 1612/4885GAA 263/4885LMNA 2845/4885
US-11702401-B2 Compounds and methods of use TGFB2, TGFB1, HDGF SMN1; SMN2 1612/4885GAA 263/4885LMNA 2845/4885
US-20130196927-A1 Smac Mimetic Therapy BIRC7, BIRC2, BIRC3 SMN1; SMN2 76/4885GAA 2299/4885LMNA 676/4885
US-20140303090-A1 Smac Mimetic Therapy XIAP, BIRC3, BIRC5 SMN1; SMN2 38/4885GAA 3080/4885LMNA 210/4885
US-11053216-B2 Compounds and methods of use TGFB2, TGFB1, HDGF SMN1; SMN2 1612/4885GAA 263/4885LMNA 2845/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.