SCHEMBL19339591

SCHEMBL19339591

CCCN(Cc1nc2ccc(Br)cc2[nH]1)C(=O)OC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC11 Q96DB2 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
HDAC9 Q9UKV0 1/20 0.43
HDAC5 Q9UQL6 1/20 0.43
DRD1 P21728 1/20 0.40
EGFR P00533 1/20 0.40
CACNA1G O43497 3/20 0.39
CACNA1B Q00975 1/20 0.39
CACNA1C Q13936 1/20 0.39
MMP2 P08253 2/20 0.39
MMP9 P14780 2/20 0.39
MMP8 P22894 2/20 0.39
MMP13 P45452 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10201483 0.92 CACNA1G (0.39) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL19488323 0.86 NPSR1 (0.51) HDAC6CACNA1GCACNA1BCACNA1CALDH1A1
SCHEMBL19883604 0.85 LMNA (0.37) HDAC3HDAC1HDAC2CACNA1GCACNA1B
SCHEMBL19488867 0.85 KDM4E (0.48) HDAC3HDAC1HDAC2MMP2MMP9
SCHEMBL19339742 0.85 GABRA1 (0.39) HDAC3HDAC1HDAC2HDAC6CACNA1G
SCHEMBL19488634 0.84 NPSR1 (0.38) HDAC3HDAC1HDAC2CACNA1GCACNA1B
SCHEMBL19488842 0.84 NPSR1 (0.38) HDAC3HDAC1HDAC2HDAC6CACNA1G
SCHEMBL10200220 0.81 CACNA1G (0.39) HDAC3HDAC1HDAC2CACNA1GCACNA1B
SCHEMBL10202452 0.78 GABRA1 (0.41) HDAC3HDAC1HDAC2CACNA1GCACNA1B
SCHEMBL19488627 0.78 ALDH1A1 (0.48) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3002281-B1 ANTIVIRAL COMPOUNDS GILEAD PHARMASSET LLC (US) 2017-09-13 EP disclosed