SCHEMBL19360299

SCHEMBL19360299

COC(=O)c1ccc2c(c1)cc(Cc1ccccc1OC)n2C(C)C

nearest known ligand 0.65

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RORC P51449 9/20 0.65
GNRHR P30968 2/20 0.42
IDH1 O75874 1/20 0.42
TP53 P04637 2/20 0.41
LMNA P02545 2/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.40
PLA2G2A P14555 1/20 0.40
HIF1A Q16665 1/20 0.40
KIF11 P52732 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19360300 0.90 RORC (0.63) RORCIDH1
SCHEMBL19360374 0.89 RORC (0.61) RORCKIF11
SCHEMBL19360367 0.89 RORC (0.66) RORCIDH1KIF11
SCHEMBL19360580 0.85 RORC (0.63) RORCKIF11
SCHEMBL19360363 0.78 RORC (0.65) RORCIDH1
SCHEMBL19360322 0.76 RORC (0.49) RORCIDH1KIF11
SCHEMBL19360371 0.76 RORC (0.62) RORCLMNA
SCHEMBL19360575 0.76 RORC (0.65) RORCKIF11
SCHEMBL19360378 0.75 RORC (0.64) RORCIDH1
SCHEMBL22004147 0.73 ACLY (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017157332-A1 AROMATIC AMIDE DERIVATIVE, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL APPLICATIONS THEREOF 江苏恒瑞医药股份有限公司 2017-09-21 WO disclosed