SCHEMBL19360613

SCHEMBL19360613

CCOC(=O)c1ccc2[nH]c(CN3CCC(C(F)(F)F)CC3)cc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.44
BCHE P06276 1/20 0.44
MAOA P21397 1/20 0.44
ACHE P22303 1/20 0.44
MAOB P27338 1/20 0.44
MMP2 P08253 1/20 0.43
MMP13 P45452 1/20 0.43
ALDH1A1 P00352 6/20 0.42
MEN1 O00255 5/20 0.42
KMT2A Q03164 5/20 0.42
MAPK1 P28482 3/20 0.42
MAPT P10636 3/20 0.42
CRHBP P24387 1/20 0.42
CRHR2 Q13324 1/20 0.42
HCRTR1 O43613 2/20 0.41
KDM4E B2RXH2 6/20 0.40
HSD17B10 Q99714 4/20 0.40
POLB P06746 3/20 0.40
ALOX15 P16050 1/20 0.40
RAB9A P51151 5/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28797800 0.82 MMP2 (0.43) HRH3MMP2MMP13ALDH1A1MEN1
SCHEMBL29654096 0.82 MMP2 (0.43) HRH3MMP2MMP13ALDH1A1MEN1
SCHEMBL19360625 0.77 USP2 (0.39) MAOAALDH1A1MAPK1KDM4E
SCHEMBL29654185 0.74 HRH3 (0.59) HRH3MMP2MMP13ALDH1A1MEN1
SCHEMBL5793708 0.74 KDM4E (0.57) HRH3ALDH1A1MEN1KMT2AMAPK1
SCHEMBL18440835 0.73 KDM4E (0.41) ALDH1A1MEN1KMT2AKDM4EHSD17B10
SCHEMBL7920888 0.72 ALDH1A1 (0.68) HRH3MMP2MMP13ALDH1A1MEN1
SCHEMBL10272098 0.72 HRH3 (0.47) HRH3ALDH1A1MAPTKDM4EHSD17B10
SCHEMBL18440581 0.72 HRH3 (0.48) HRH3MAOBMMP2MMP13ALDH1A1
SCHEMBL21985665 0.70 KDM4E (0.47) HRH3MMP2MMP13ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107531679-B Aromatic amide derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2021-07-02 CN disclosed
WO-2017157332-A1 AROMATIC AMIDE DERIVATIVE, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL APPLICATIONS THEREOF 江苏恒瑞医药股份有限公司 2017-09-21 WO disclosed