SCHEMBL1937548

SCHEMBL1937548

CCCCCNc1nc(Cl)ncc1Cl

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
STK17A Q9UEE5 15/20 0.54
STK17B O94768 11/20 0.54
NPSR1 Q6W5P4 2/20 0.43
KDM4E B2RXH2 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
KMT2A Q03164 1/20 0.43
S1PR2 O95136 1/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TLR8 Q9NR97 1/20 0.40
CNR2 P34972 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1937398 0.95 STK17A (0.56) STK17ASTK17BNPSR1KDM4EL3MBTL1
SCHEMBL1934538 0.88 STK17A (0.51) STK17ASTK17BL3MBTL1KMT2A
SCHEMBL25669146 0.85 STK17A (0.48) STK17ASTK17BNPSR1KDM4EL3MBTL1
SCHEMBL4188949 0.84 KMT2A (0.47) STK17ASTK17BNPSR1KDM4EL3MBTL1
SCHEMBL25584087 0.84 KMT2A (0.44) STK17ASTK17BNPSR1KDM4EL3MBTL1
SCHEMBL4194117 0.84 TLR8 (0.44) STK17ASTK17BNPSR1KDM4EL3MBTL1
SCHEMBL20154842 0.83 STK17A (0.60) STK17ASTK17B
SCHEMBL1400319 0.81 STK17A (0.56) STK17ASTK17BKMT2ALMNASMN1; SMN2
SCHEMBL20652148 0.81 STK17A (0.52) STK17ASTK17BL3MBTL1
SCHEMBL1935303 0.80 STK17B (0.47) STK17ASTK17BL3MBTL1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10774092-B2 ULK1 inhibitors and methods using same SALK INSTITUTE FOR BIOLOGICAL STUDIES (US) 2020-09-15 US disclosed
US-10689397-B2 ULK1 inhibitors and methods using same SALK INSTITUTE FOR BIOLOGICAL STUDIES (US) 2020-06-23 US disclosed
US-20190284207-A1 NOVEL ULK1 INHIBITORS AND METHODS USING SAME SALK INSTITUTE FOR BIOLOGICAL STUDIES 2019-09-19 US disclosed
US-20190248806-A1 NOVEL ULK1 INHIBITORS AND METHODS USING SAME SALK INSTITUTE FOR BIOLOGICAL STUDIES 2019-08-15 US disclosed
US-20190152989-A1 NOVEL ULK1 INHIBITORS AND METHODS USING SAME SALK INSTITUTE FOR BIOLOGICAL STUDIES 2019-05-23 US disclosed
US-10266549-B2 ULK1 inhibitors and methods using same SALK INSTITUTE FOR BIOLOGICAL STUDIES (US) 2019-04-23 US disclosed
US-20170342088-A1 NOVEL ULK1 INHIBITORS AND METHODS USING SAME SALK INSTITUTE FOR BIOLOGICAL STUDIES (US) 2017-11-30 US disclosed
EP-3185868-A1 NOVEL ULK1 INHIBITORS AND METHODS USING SAME Salk Institute for Biological Studies (US) 2017-07-05 EP disclosed
WO-2016033100-A1 NOVEL ULK1 INHIBITORS AND METHODS USING SAME SALK INSTITUTE FOR BIOLOGICAL STUDIES (US) 2016-03-03 WO disclosed
US-20110230478-A1 4-Alkyl-substituted diaminopyrimidines Bayer ScienceCrop AG (DE) 2011-09-22 US disclosed
EP-2330904-A2 4-ALKYL-SUBSTITUTED DIAMINOPYRIMIDINES Bayer CropScience AG (DE) 2011-06-15 EP disclosed
WO-2010025863-A2 4-ALKYL-SUBSTITUTED DIAMINOPYRIMIDINES BAYER CROPSCIENCE AG (DE) 2010-03-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10689397-B2 ULK1 inhibitors and methods using same ULK1, ULK2, ULK3 STK17A 68/4885STK17B 129/4885NPSR1 4371/4885
US-10266549-B2 ULK1 inhibitors and methods using same ULK1, ULK2, ULK3 STK17A 68/4885STK17B 129/4885NPSR1 4371/4885
US-20170342088-A1 NOVEL ULK1 INHIBITORS AND METHODS USING SAME ULK1, ULK2, ULK3 STK17A 69/4885STK17B 116/4885NPSR1 4283/4885
US-20110230478-A1 4-Alkyl-substituted diaminopyrimidines DPM1, DPYD, POLR1C STK17A 2888/4885STK17B 3187/4885NPSR1 4180/4885
US-20190248806-A1 NOVEL ULK1 INHIBITORS AND METHODS USING SAME ULK1, ULK2, ULK3 STK17A 69/4885STK17B 116/4885NPSR1 4283/4885
US-20190152989-A1 NOVEL ULK1 INHIBITORS AND METHODS USING SAME ULK1, ULK2, ULK3 STK17A 69/4885STK17B 116/4885NPSR1 4283/4885
US-10774092-B2 ULK1 inhibitors and methods using same ULK1, ULK2, ULK3 STK17A 68/4885STK17B 129/4885NPSR1 4371/4885
US-20190284207-A1 NOVEL ULK1 INHIBITORS AND METHODS USING SAME ULK1, ULK2, ULK3 STK17A 69/4885STK17B 116/4885NPSR1 4283/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.