SCHEMBL19386255

SCHEMBL19386255

CCCCc1nc(O)c(C(=O)OCCCc2ccccc2)c(=O)[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.47
MMP1 P03956 1/20 0.44
MMP2 P08253 1/20 0.44
MMP12 P39900 1/20 0.44
RNASEH1 O60930 2/20 0.43
ALDH1A1 P00352 4/20 0.42
MAPK1 P28482 2/20 0.42
CYP3A4 P08684 1/20 0.42
TSHR P16473 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
LMNA P02545 2/20 0.41
DAO P14920 1/20 0.41
HCAR2 Q8TDS4 1/20 0.41
NAAA Q02083 2/20 0.41
MEN1 O00255 1/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7323966 0.77 PARP1 (0.56) PARP1RNASEH1ALDH1A1TSHRL3MBTL1
SCHEMBL15271657 0.70 TSHR (0.54) ALDH1A1MAPK1CYP3A4TSHRTDP1
SCHEMBL26688876 0.70 ALDH1A1 (0.46) PARP1ALDH1A1TSHRLMNAMAPT
SCHEMBL9126680 0.69 PARP1 (0.56) PARP1RNASEH1ALDH1A1CYP3A4TSHR
SCHEMBL2018005 0.68 LMNA (0.62) ALDH1A1MAPK1CYP3A4TSHRTDP1
Butylbenzyl SCHEMBL27296811 0.68 ALDH1A1 (0.79) ALDH1A1MAPK1CYP3A4TSHRTDP1
SCHEMBL2021418 0.67 LMNA (0.60) ALDH1A1MAPK1CYP3A4TSHRTDP1
Hexane SCHEMBL28355428 0.67 LMNA (0.60) ALDH1A1MAPK1CYP3A4TSHRTDP1
SCHEMBL7323950 0.67 PARP1 (0.56) PARP1RNASEH1ALDH1A1LMNADAO
SCHEMBL20656207 0.67 MMP2 (0.47) MMP1MMP2MMP12ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3433247-A1 6-HYDROXY-4-OXO-1,4-DIHYDROPYRIMIDINE-5-CARBOXAMIDES AS APJ AGONISTS Bristol-Myers Squibb Company (US) 2019-01-30 EP disclosed
WO-2017165640-A1 6-HYDROXY-4-OXO-1,4-DIHYDROPYRIMIDINE-5-CARBOXAMIDES AS APJ AGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2017-09-28 WO disclosed