SCHEMBL19425952

SCHEMBL19425952

c1ccc2[nH]c(-c3ccc4[nH]c(-c5ccc6ocnc6c5)nc4c3)cc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FOXO1 Q12778 1/20 0.44
NPC1 O15118 12/20 0.41
RAB9A P51151 12/20 0.41
DYRK1A Q13627 1/20 0.41
KDM4E B2RXH2 8/20 0.41
ALDH1A1 P00352 6/20 0.41
MAPT P10636 5/20 0.41
HPGD P15428 4/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
CASP3 P42574 2/20 0.41
SENP8 Q96LD8 2/20 0.41
SENP7 Q9BQF6 2/20 0.41
SENP6 Q9GZR1 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
ESR1 P03372 1/20 0.41
SMN1; SMN2 Q16637 6/20 0.39
POLB P06746 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18671143 0.92 ESR1 (0.43) FOXO1NPC1RAB9ADYRK1AKDM4E
SCHEMBL19287942 0.92 ESR1 (0.48) FOXO1NPC1RAB9ADYRK1AKDM4E
SCHEMBL19155375 0.85 RIPK1 (0.46) FOXO1
SCHEMBL19557533 0.85 NPC1 (0.53) FOXO1NPC1RAB9ADYRK1AKDM4E
SCHEMBL18880102 0.84 ESR1 (0.49) NPC1RAB9ADYRK1AKDM4EALDH1A1
SCHEMBL21966181 0.81 DYRK1A (0.41) FOXO1NPC1RAB9ADYRK1AKDM4E
SCHEMBL20022978 0.81 DYRK1A (0.43) FOXO1NPC1RAB9ADYRK1AKDM4E
SCHEMBL21099202 0.80 NPC1 (0.50) NPC1RAB9ADYRK1AKDM4EALDH1A1
SCHEMBL23507947 0.79 DYRK1A (0.39) FOXO1NPC1RAB9ADYRK1AKDM4E
SCHEMBL21298764 0.78 RIPK1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11530175-B2 Method for preparation of fluoro alkylated compounds by homogeneous Ni catalysis ARXADA AG (CH) 2022-12-20 US disclosed
US-20220041530-A1 Method for Preparation of Fluoro Alkylated Compounds by Homogeneous NI Catalysis LONZA LTD (CH) 2022-02-10 US disclosed
US-10183012-B2 Compounds and compositions and methods of use ARDEA BIOSCIENCES, INC. (US) 2019-01-22 US disclosed
US-20170281601-A1 NOVEL COMPOUNDS AND COMPOSITIONS AND METHODS OF USE ARDEA BIOSCIENCES, INC. 2017-10-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220041530-A1 Method for Preparation of Fluoro Alkylated Compounds by Homogeneous NI Catalysis ABL1, AFF2, NAF1 FOXO1 3292/4885NPC1 329/4885RAB9A 655/4885
US-11530175-B2 Method for preparation of fluoro alkylated compounds by homogeneous Ni catalysis ABL1, AFF2, NAF1 FOXO1 3292/4885NPC1 329/4885RAB9A 655/4885
US-10183012-B2 Compounds and compositions and methods of use XDH, PON1, OAT FOXO1 2730/4885NPC1 732/4885RAB9A 3068/4885
US-20170281601-A1 NOVEL COMPOUNDS AND COMPOSITIONS AND METHODS OF USE XDH, PON1, GLS FOXO1 2364/4885NPC1 561/4885RAB9A 2885/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.