SCHEMBL19447299

SCHEMBL19447299

CCc1cc2c(OC(F)F)cccc2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 5/20 0.44
MTNR1B P49286 5/20 0.44
RHEB Q15382 3/20 0.44
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
PARP1 P09874 1/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
ATM Q13315 1/20 0.37
NR3C1 P04150 4/20 0.36
PGR P06401 3/20 0.36
NR3C2 P08235 3/20 0.36
FLT3 P36888 1/20 0.35
ABCB11 O95342 1/20 0.34
HTR1A P08908 1/20 0.34
ADRA2A P08913 1/20 0.34
PTGS1 P23219 1/20 0.34
SLC6A2 P23975 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25267 0.81 MTNR1A (0.62) MTNR1AMTNR1BRHEBHDAC3HDAC1
SCHEMBL24451623 0.80 MTNR1A (0.45) MTNR1AMTNR1BRHEBPARP1MEN1
SCHEMBL12475578 0.80 HTR1A (0.48) RHEBHDAC3HDAC1MEN1NPC1
SCHEMBL24459343 0.79 MTNR1A (0.45) MTNR1AMTNR1BRHEBPARP1MEN1
SCHEMBL10377783 0.78 MTNR1A (0.42) MTNR1AMTNR1BRHEBPARP1MEN1
SCHEMBL20097158 0.78 RHEB (0.56) MTNR1AMTNR1BRHEBABCB11HTR1A
SCHEMBL15077049 0.77 MEN1 (0.38) MTNR1AMTNR1BRHEBHDAC3HDAC1
SCHEMBL30304098 0.74 KDM4E (0.49) HDAC3HDAC1MEN1NPC1RAB9A
SCHEMBL17345632 0.74 DAO (0.49) MTNR1AMTNR1BRHEBPARP1FLT3
SCHEMBL5768529 0.74 SRD5A2 (0.61) MTNR1AMTNR1BRHEBHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2794611-B1 PYRAZOLO[1,5-A]PYRIMIDINES AS ANTIVIRAL AGENTS GILEAD SCIENCES INC (US) 2017-10-11 EP disclosed