SCHEMBL19475326

SCHEMBL19475326

Nc1ccc(-c2cc(CN3CCOCC3)c3cccc(Cl)c3n2)nc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 3/20 0.50
RAB9A P51151 2/20 0.50
NPC1 O15118 1/20 0.50
PAX8 Q06710 1/20 0.50
MOK Q9UQ07 7/20 0.48
METAP2 P50579 1/20 0.45
CYP2A13 Q16696 5/20 0.44
SMN1; SMN2 Q16637 3/20 0.40
MAPT P10636 3/20 0.40
HTT P42858 2/20 0.40
KDM4E B2RXH2 2/20 0.40
LMNA P02545 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
POLB P06746 1/20 0.40
MCL1 Q07820 1/20 0.40
MAP4K4 O95819 1/20 0.38
ALOX5AP P20292 1/20 0.38
FEN1 P39748 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19475290 0.86 MOK (0.52) L3MBTL1RAB9ANPC1PAX8MOK
SCHEMBL19475395 0.84 MOK (0.66) MOKMAPTKDM4ELMNATDP1
SCHEMBL19475494 0.81 MOK (0.76) MOK
SCHEMBL19475304 0.80 MOK (0.73) MOKKDM4ELMNAPOLB
SCHEMBL14988278 0.72 NCF1 (0.53) HTTKDM4EMAP4K4
SCHEMBL19475283 0.72 MOK (0.75) MOK
SCHEMBL19475336 0.69 MOK (0.67) L3MBTL1RAB9ANPC1MOKMAPT
SCHEMBL19475402 0.69 HAVCR2 (0.55) RAB9ANPC1MOKMAPTHTT
SCHEMBL31590658 0.69 MOK (0.55) MOKCYP2A13KDM4E
SCHEMBL27253776 0.67 L3MBTL1 (1.00) L3MBTL1RAB9ANPC1PAX8METAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11192859-B2 Quinoline compounds as modulators of RAGE activity and uses thereof UNIV NEW YORK (US) 2021-12-07 US disclosed
US-11192859-B2 Quinoline compounds as modulators of RAGE activity and uses thereof UNIV NEW YORK (US) 2021-12-07 US disclosed
US-20190194136-A1 QUINOLINE COMPOUNDS AS MODULATORS OF RAGE ACTIVITY AND USES THEREOF UNIV NEW YORK (US) 2019-06-27 US disclosed
US-20190194136-A1 QUINOLINE COMPOUNDS AS MODULATORS OF RAGE ACTIVITY AND USES THEREOF UNIV NEW YORK (US) 2019-06-27 US disclosed
WO-2017184547-A1 QUINOLINE COMPOUNDS AS MODULATORS OF RAGE ACTIVITY AND USES THEREOF NEW YORK UNIVERSITY (US) 2017-10-26 WO disclosed
WO-2017184547-A1 QUINOLINE COMPOUNDS AS MODULATORS OF RAGE ACTIVITY AND USES THEREOF NEW YORK UNIVERSITY (US) 2017-10-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190194136-A1 QUINOLINE COMPOUNDS AS MODULATORS OF RAGE ACTIVITY AND USES THEREOF AGER, HMGB1, GPR119 L3MBTL1 2976/4885RAB9A 1174/4885NPC1 3452/4885
US-11192859-B2 Quinoline compounds as modulators of RAGE activity and uses thereof AGER, HMGB1, GPR119 L3MBTL1 2976/4885RAB9A 1174/4885NPC1 3452/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.