SCHEMBL19476138

SCHEMBL19476138

O=C(Nc1ccccc1-c1ccccc1)c1cscn1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.63
TSHR P16473 4/20 0.63
ALOX15 P16050 1/20 0.63
PIM1 P11309 1/20 0.56
KDM4E B2RXH2 3/20 0.55
ATM Q13315 1/20 0.55
L3MBTL1 Q9Y468 2/20 0.54
GRM1 Q13255 1/20 0.51
HSD17B10 Q99714 2/20 0.50
LMNA P02545 1/20 0.50
MAPT P10636 2/20 0.48
HTT P42858 2/20 0.48
USP2 O75604 1/20 0.48
POLB P06746 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
IRAK4 Q9NWZ3 1/20 0.46
GRM4 Q14833 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19476100 0.82 TSHR (0.74) ALDH1A1TSHRALOX15KDM4EATM
SCHEMBL26627433 0.79 PIM1 (0.59) ALDH1A1PIM1KDM4EGRM1MEN1
SCHEMBL13626622 0.79 PIM1 (0.59) ALDH1A1PIM1KDM4EGRM1HSD17B10
SCHEMBL6287453 0.79 HDAC1 (0.68) ALDH1A1PIM1GRM1GRM4
SCHEMBL168520 0.79 GRM4 (0.63) ALDH1A1PIM1KDM4EGRM1POLB
Ammonia Solution, Strong SCHEMBL27976383 0.78 PIM1 (0.57) ALDH1A1PIM1KDM4EGRM1HSD17B10
SCHEMBL1034502 0.77 PIM1 (0.48) ALDH1A1TSHRALOX15PIM1KDM4E
SCHEMBL19476101 0.77 TSHR (0.65) ALDH1A1TSHRPIM1ATML3MBTL1
SCHEMBL12666639 0.76 PIM1 (0.55) ALDH1A1PIM1KDM4EATML3MBTL1
SCHEMBL20541724 0.76 SIRT1 (0.66) ALDH1A1TSHRALOX15KDM4EATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10759765-B2 Heterocyclic carboxylic acid amide ligand and applications thereof in copper catalyzed coupling reaction of aryl halogeno substitute CE PHARM CO., LTD. (CN) 2020-09-01 US disclosed
US-20190127337-A1 HETEROCYCLIC CARBOXYLIC ACID AMIDE LIGAND AND APPLICATIONS THEREOF IN COPPER CATALYZED COUPLING REACTION OF ARYL HALOGENO SUBSTITUTE CE PHARM CO., LTD. (CN) 2019-05-02 US disclosed
WO-2017177979-A1 HETEROCYCLIC CARBOXYLIC ACID AMIDE LIGAND AND APPLICATIONS THEREOF IN COPPER CATALYZED COUPLING REACTION OF ARYL HALOGENO SUBSTITUTE 中国科学院上海有机化学研究所 2017-10-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190127337-A1 HETEROCYCLIC CARBOXYLIC ACID AMIDE LIGAND AND APPLICATIONS THEREOF IN COPPER CATALYZED COUPLING REACTION OF ARYL HALOGENO SUBSTITUTE AOC1, AOC2, AOC3 ALDH1A1 79/4885TSHR 190/4885ALOX15 312/4885
US-10759765-B2 Heterocyclic carboxylic acid amide ligand and applications thereof in copper catalyzed coupling reaction of aryl halogeno substitute AOC1, AOC2, AOC3 ALDH1A1 79/4885TSHR 190/4885ALOX15 312/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.