SCHEMBL19476173

SCHEMBL19476173

O=S(=O)(c1ccccc1)c1ccc2sccc2c1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA12 O43570 5/20 0.54
CA2 P00918 5/20 0.54
HTR6 P50406 5/20 0.48
CTNNB1 P35222 1/20 0.45
WNT3A P56704 1/20 0.45
PIK3CD O00329 1/20 0.44
ALDH1A1 P00352 1/20 0.44
POLB P06746 1/20 0.44
MAPT P10636 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CYP2A6 P11509 1/20 0.43
PTPRC P08575 1/20 0.43
PTPN6 P29350 1/20 0.43
PTPN11 Q06124 1/20 0.43
PTPN22 Q9Y2R2 1/20 0.43
NPSR1 Q6W5P4 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6234706 0.78 CA2 (0.80) CA12CA2SMN1; SMN2
SCHEMBL6737344 0.77 CA2 (0.51) CA12CA2CYP2A6PTPRCPTPN6
SCHEMBL4231613 0.77 CA2 (0.51) CA12CA2CYP2A6PTPRCPTPN6
SCHEMBL6378197 0.77 CYP2A6 (0.47) CA12CA2HTR6PIK3CDALDH1A1
SCHEMBL3793170 0.77 CYP2A6 (0.47) CA12CA2CTNNB1WNT3AALDH1A1
SCHEMBL12333390 0.74 PIK3CD (0.44) CA12CA2HTR6CTNNB1WNT3A
SCHEMBL3934050 0.74 HTR6 (0.61) CA2HTR6ALDH1A1POLBMAPT
SCHEMBL3795030 0.72 CA2 (0.51) CA12CA2HTR6CYP2A6PTPRC
SCHEMBL5051390 0.72 HTR6 (0.93) CA12CA2HTR6ALDH1A1POLB
SCHEMBL8371819 0.70 IKBKB (0.48) HTR6PIK3CDALDH1A1POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10759765-B2 Heterocyclic carboxylic acid amide ligand and applications thereof in copper catalyzed coupling reaction of aryl halogeno substitute CE PHARM CO., LTD. (CN) 2020-09-01 US disclosed
US-20190127337-A1 HETEROCYCLIC CARBOXYLIC ACID AMIDE LIGAND AND APPLICATIONS THEREOF IN COPPER CATALYZED COUPLING REACTION OF ARYL HALOGENO SUBSTITUTE CE PHARM CO., LTD. (CN) 2019-05-02 US disclosed
WO-2017177979-A1 HETEROCYCLIC CARBOXYLIC ACID AMIDE LIGAND AND APPLICATIONS THEREOF IN COPPER CATALYZED COUPLING REACTION OF ARYL HALOGENO SUBSTITUTE 中国科学院上海有机化学研究所 2017-10-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190127337-A1 HETEROCYCLIC CARBOXYLIC ACID AMIDE LIGAND AND APPLICATIONS THEREOF IN COPPER CATALYZED COUPLING REACTION OF ARYL HALOGENO SUBSTITUTE AOC1, AOC2, AOC3 CA12 470/4885CA2 743/4885HTR6 3576/4885
US-10759765-B2 Heterocyclic carboxylic acid amide ligand and applications thereof in copper catalyzed coupling reaction of aryl halogeno substitute AOC1, AOC2, AOC3 CA12 470/4885CA2 743/4885HTR6 3576/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.