SCHEMBL19518992

SCHEMBL19518992

CC(C)(O)c1ccc(S(=O)(=O)NC(=O)Nc2c3c(c(Cl)c4c2CCC4)CCC3)cc1

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 12/20 0.54
CA2 P00918 2/20 0.51
CA1 P00915 1/20 0.46
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24592610 0.92 NLRP3 (0.58) NLRP3CA2CA1KMT2A
SCHEMBL19518993 0.88 NLRP3 (0.54) NLRP3CA2KMT2A
SCHEMBL19519058 0.87 NLRP3 (0.66) NLRP3CA2
SCHEMBL19519040 0.86 NLRP3 (0.74) NLRP3CA2
SCHEMBL19475370 0.85 NLRP3 (0.54) NLRP3CA2
SCHEMBL19519054 0.85 NLRP3 (0.51) NLRP3CA2KMT2A
SCHEMBL23378793 0.84 GSTO1 (0.52) NLRP3CA2
SCHEMBL19518977 0.83 NLRP3 (0.49) NLRP3CA2
SCHEMBL23957303 0.82 NLRP3 (0.50) NLRP3CA2
SCHEMBL23378794 0.82 NLRP3 (0.48) NLRP3CA2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11597706-B2 Compounds and compositions for treating conditions associated with NLRP activity NOVARTIS AG (CH) 2023-03-07 US disclosed
US-11597706-B2 Compounds and compositions for treating conditions associated with NLRP activity NOVARTIS AG (CH) 2023-03-07 US disclosed
EP-3445756-B1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2022-07-06 EP disclosed
US-20190119203-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2019-04-25 US disclosed
US-20190119203-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2019-04-25 US disclosed
WO-2017184623-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY IFM THERAPEUTICS, INC (US) 2017-10-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11597706-B2 Compounds and compositions for treating conditions associated with NLRP activity NLRP1, NLRP3, NOD1 NLRP3 2/4885CA2 2191/4885CA1 4294/4885
US-20190119203-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NLRP1, NLRP3, NOD1 NLRP3 2/4885CA2 2191/4885CA1 4294/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.