SCHEMBL19554186

SCHEMBL19554186

COc1cc(NC(=O)c2ccc3cc(C(F)(F)F)ccc3c2)c(C(=O)O)cc1C#N

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.48
KDM4E B2RXH2 3/20 0.47
AKR1C4 P17516 1/20 0.46
AKR1C3 P42330 1/20 0.46
AKR1C2 P52895 1/20 0.46
AKR1C1 Q04828 1/20 0.46
PLK1 P53350 1/20 0.46
KCNK2 O95069 2/20 0.45
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2C19 P33261 2/20 0.45
CYP2D6 P10635 1/20 0.45
KCNK10 P57789 1/20 0.45
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA7 P43166 1/20 0.45
TAS2R14 Q9NYV8 1/20 0.45
MAPK1 P28482 1/20 0.45
KMT2A Q03164 2/20 0.44
CYP2C9 P11712 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19554219 0.87 AKR1C4 (0.48) MAPTKDM4EAKR1C4AKR1C3AKR1C2
SCHEMBL19554333 0.87 AKR1C4 (0.56) MAPTKDM4EAKR1C4AKR1C3AKR1C2
SCHEMBL19554329 0.85 MAPT (0.59) MAPTKDM4EAKR1C4AKR1C3AKR1C2
SCHEMBL19554266 0.85 KMT2A (0.55) MAPTKDM4EAKR1C4AKR1C3AKR1C2
SCHEMBL19554216 0.78 AKR1C4 (0.46) MAPTKDM4EAKR1C4AKR1C3AKR1C2
SCHEMBL19554239 0.77 MAPT (0.49) MAPTKDM4EAKR1C4AKR1C3AKR1C2
SCHEMBL19554178 0.77 NPC1 (0.52) KDM4EAKR1C2AKR1C1CYP1A2CYP3A4
SCHEMBL19570245 0.74 NPC1 (0.49) MAPTKDM4EAKR1C2AKR1C1CYP1A2
SCHEMBL19554188 0.74 F11 (0.47) AKR1C4AKR1C3AKR1C2AKR1C1CA12
SCHEMBL19554253 0.74 F11 (0.46) MAPTAKR1C4AKR1C3AKR1C2AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO claimed
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO disclosed
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO disclosed