SCHEMBL19554231

SCHEMBL19554231

CSc1cc(NC(=O)c2ccc3cc(Cl)ccc3c2)c(C(=O)O)cc1C#N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.50
MEN1 O00255 4/20 0.50
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
PKM P14618 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
SERPINE1 P05121 5/20 0.45
AKR1C4 P17516 1/20 0.43
AKR1C3 P42330 1/20 0.43
AKR1C2 P52895 1/20 0.43
AKR1C1 Q04828 1/20 0.43
KCNK2 O95069 2/20 0.43
KCNK10 P57789 2/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19554190 0.86 KMT2A (0.49) KMT2AMEN1PKMNPSR1SERPINE1
SCHEMBL19554136 0.86 MEN1 (0.48) KMT2AMEN1PKMNPSR1SERPINE1
SCHEMBL19554266 0.83 KMT2A (0.55) KMT2AMEN1PKMNPSR1SERPINE1
SCHEMBL19554218 0.83 MEN1 (0.47) KMT2AMEN1PKMNPSR1SERPINE1
SCHEMBL19554236 0.82 SERPINE1 (0.46) KMT2AMEN1PKMNPSR1SERPINE1
SCHEMBL19570245 0.81 NPC1 (0.49) KMT2AMEN1CYP1A2CYP3A4PKM
SCHEMBL19554188 0.81 F11 (0.47) KMT2AMEN1PKMNPSR1SERPINE1
SCHEMBL19554253 0.79 F11 (0.46) KMT2AMEN1PKMNPSR1SERPINE1
SCHEMBL19554161 0.78 CA2 (0.56) KMT2AMEN1SERPINE1AKR1C4AKR1C3
SCHEMBL19554134 0.77 SERPINE1 (0.68) SERPINE1AKR1C4AKR1C3AKR1C2AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO claimed
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO disclosed
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO disclosed