SCHEMBL19558166

SCHEMBL19558166

CC(C)(C)Nc1ccc(-c2nn[nH]n2)cc1

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
XDH P47989 9/20 0.60
ADH5 P11766 1/20 0.60
TP53 P04637 3/20 0.57
RPA1 P27694 1/20 0.53
ATM Q13315 1/20 0.53
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
ALDH1A1 P00352 2/20 0.53
CYP19A1 P11511 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
GPR35 Q9HC97 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16144653 0.80 ADH5 (0.67) XDHADH5TP53RPA1ATM
SCHEMBL9984638 0.79 ADH5 (0.95) XDHADH5TP53RPA1ATM
SCHEMBL3413673 0.77 XDH (0.96) XDHADH5TP53RPA1ATM
SCHEMBL14381411 0.77 ADH5 (0.67) XDHADH5TP53RPA1ATM
SCHEMBL23987210 0.75 XDH (0.68) XDHADH5TP53RPA1ATM
SCHEMBL2667739 0.74 ADH5 (0.75) XDHADH5TP53RPA1ATM
SCHEMBL15004536 0.73 MAPT (0.69) XDHADH5TP53ALDH1A1GPR35
SCHEMBL1344194 0.73 TP53 (1.00) XDHADH5TP53RPA1ATM
SCHEMBL18896243 0.72 ADH5 (0.60) XDHADH5TP53RPA1ATM
SCHEMBL9969399 0.72 TP53 (0.67) XDHADH5TP53RPA1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9809545-B2 Factor XIa inhibitors MERCK SHARP & DOHME CORP. (US) 2017-11-07 US disclosed