SCHEMBL1957955

SCHEMBL1957955

COc1ccccc1-c1ccccc1CC=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 4/20 0.46
ALDH1A1 P00352 3/20 0.45
CHRM2 P08172 3/20 0.44
CHRM1 P11229 2/20 0.44
CHRM3 P20309 1/20 0.44
APP P05067 1/20 0.43
GAA P10253 1/20 0.42
ERN1 O75460 1/20 0.42
IDO1 P14902 2/20 0.42
TAAR1 Q96RJ0 1/20 0.42
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
HPGD P15428 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4746229 0.87 MEN1 (0.43) ALDH1A1CHRM2CHRM1CHRM3GAA
SCHEMBL249539 0.85 ALDH1A1 (0.54) ALDH1A1CHRM2CHRM1CHRM3IDO1
SCHEMBL29957820 0.85 ALDH1A1 (0.54) ALDH1A1CHRM2CHRM1CHRM3IDO1
SCHEMBL14894360 0.83 SLC22A12 (0.48) ALDH1A1GAAHPGDCYP1A2CYP3A4
SCHEMBL5045738 0.83 CHRM2 (0.45) HTR7ALDH1A1CHRM2CHRM1CHRM3
SCHEMBL1515714 0.79 L3MBTL1 (0.46) HTR7ALDH1A1GAAERN1HPGD
SCHEMBL19043338 0.77 SLC13A5 (0.49) HTR7ALDH1A1ERN1HPGD
SCHEMBL5205282 0.76 CA12 (0.49) ALDH1A1GAACA12CA1CA2
SCHEMBL6177247 0.76 ALDH1A1 (0.47) ALDH1A1CHRM2CHRM1CHRM3IDO1
SCHEMBL1515689 0.76 ABL1 (0.50) HTR7IDO1CYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2507215-A1 DIPHENYL AZEPINE DERIVATIVES AS MONOAMINE REUPTAKE INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-10-10 EP disclosed
WO-2011067219-A1 DIPHENYL AZEPINE DERIVATIVES AS MONOAMINE REUPTAKE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2011-06-09 WO disclosed